SCHEMBL16601602

SCHEMBL16601602

CCN1C(=O)C2(CCC2)Oc2cc(C)ccc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 2/20 0.40
POLB P06746 1/20 0.39
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 3/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.35
ALPL P05186 1/20 0.35
ATM Q13315 1/20 0.35
F2 P00734 1/20 0.34
GAA P10253 1/20 0.34
ALOX12 P18054 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13367654 0.90 NR3C2 (0.39) NR3C2POLBALDH1A1MAPTKDM4E
SCHEMBL17434459 0.85 ATAD2 (0.44) NR3C2ALDH1A1MAPTMAPK1TDP1
SCHEMBL13961731 0.85 NR3C2 (0.39) NR3C2ALDH1A1HTTKMT2AALPL
SCHEMBL13340973 0.83 NR3C2 (0.38) NR3C2ALDH1A1MAPTKMT2ATSHR
SCHEMBL16601600 0.82 NR3C2 (0.45) NR3C2POLBALDH1A1MAPTKDM4E
SCHEMBL17434319 0.81 MAPT (0.39) NR3C2POLBALDH1A1MAPTTDP1
SCHEMBL13367651 0.80 RXRA (0.43) NR3C2POLBALDH1A1MAPTMAPK1
SCHEMBL17434414 0.80 ATAD2 (0.46) NR3C2ALDH1A1MAPTMAPK1TDP1
SCHEMBL16601592 0.79 KMT2A (0.38) POLBALDH1A1MAPTMAPK1TDP1
SCHEMBL13367760 0.78 SLC9A1 (0.40) NR3C2POLBALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8993585-B2 Cyclic amine substituted pyrimidinediamines as PKC inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-03-31 US disclosed