SCHEMBL16607648

SCHEMBL16607648

NCc1ccc(Br)cc1CC(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.40
CCR5 P51681 1/20 0.37
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SLC6A4 P31645 1/20 0.32
KDM1A O60341 2/20 0.31
HTR2A P28223 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390800 0.81 CYP2A6 (0.48) CYP2A6CCR5ALDH1A1KDM4EMEN1
SCHEMBL16609146 0.81 PTGDR2 (0.40) ALDH1A1MEN1MAPTKMT2ASLC6A4
SCHEMBL11713314 0.78 MAPT (0.38) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL31349168 0.78 ALDH1A1 (0.38) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL1055260 0.76 PYCR1 (0.44) KDM1A
SCHEMBL1823372 0.74 KDM1A (0.46) CYP2A6CCR5KDM1A
SCHEMBL31717131 0.74 KDM1A (0.46) CYP2A6CCR5KDM1A
SCHEMBL24970154 0.74 KDM1A (0.42) CYP2A6CCR5SLC6A4KDM1A
SCHEMBL3985481 0.74 TSHR (0.46) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL23094700 0.74 ALOX15 (0.40) ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015046405-A1 ANALGESIC 東レ株式会社 2015-04-02 WO disclosed
WO-2015046404-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR PULMONARY HYPERTENSION 東レ株式会社 2015-04-02 WO disclosed