SCHEMBL16615276

SCHEMBL16615276

Clc1ccc(Cl)c(CN2CCNc3c2c2c(-c4nc(C5CCCN5)no4)n3-2)c1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
EPHA2 P29317 1/20 0.31
KDR P35968 1/20 0.31
GPR6 P46095 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615265 0.88 NPC1 (0.43) ALKCHRM1CHRM3GPR6
SCHEMBL16615266 0.84 LMNA (0.38) ALKMAPTCYP2C9CYP2C19
SCHEMBL17969717 0.74 ALK (0.40) ALKCHRM1CHRM3KDR
SCHEMBL16615336 0.73 LMNA (0.35) ALKMAPTCYP2C19
SCHEMBL16615327 0.73 ALK (0.40) ALKMAPT
SCHEMBL16615324 0.72 ALK (0.34) ALK
SCHEMBL16615200 0.72 CHRM1 (0.45) CHRM1CHRM3
SCHEMBL16615312 0.70 NR1H4 (0.36)
SCHEMBL16615186 0.69 ALK (0.34) ALKGPR6
SCHEMBL17918692 0.67 NPC1 (0.42) ALKCHRM1CHRM3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed