SCHEMBL1661572

SCHEMBL1661572

Cc1nc2ccc(C3(c4ccccc4)C=C3)nc2s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 9/20 0.41
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
MAOB P27338 1/20 0.33
KMT2A Q03164 1/20 0.32
ALOX5 P09917 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCND1 P24385 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661650 0.81 S1PR1 (0.42) S1PR1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL1661570 0.81 S1PR1 (0.62) S1PR1COMT
SCHEMBL1661564 0.75 S1PR1 (0.50) S1PR1MAOBALOX5
SCHEMBL1661678 0.75 S1PR1 (0.44) S1PR1MAOB
SCHEMBL1662792 0.75 APP (0.50) S1PR1MAOB
SCHEMBL1661615 0.74 MAOB (0.40) S1PR1MAOB
SCHEMBL1661809 0.74 S1PR1 (0.39) S1PR1MAOB
SCHEMBL1661196 0.74 S1PR1 (0.39) S1PR1SMN1; SMN2NPC1HTTRAB9A
SCHEMBL1661173 0.74 ALDH1A1 (0.34) S1PR1
SCHEMBL1661097 0.74 S1PR1 (0.43) S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed