SCHEMBL16615790

SCHEMBL16615790

C=C(C)S/C(=C\C)CNC(=O)c1ccc(CNC(=O)c2cccc(C#N)c2)cn1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 10/20 0.45
GAA P10253 1/20 0.41
GPR139 Q6DWJ6 1/20 0.40
CHRM3 P20309 1/20 0.39
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
GRM5 P41594 1/20 0.38
PRKAA2 P54646 1/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615837 0.76 VNN1 (0.48) VNN1GAACHRM3ROCK2ROCK1
SCHEMBL11627692 0.69 VNN1 (0.67) VNN1ROCK2ALDH1A1
SCHEMBL7985996 0.68 GAA (0.56) VNN1GAACHRM3ALDH1A1
SCHEMBL17142140 0.68 HDAC2 (0.64) VNN1GAAGPR139CHRM3ALDH1A1
SCHEMBL7986109 0.67 MAOB (0.55) VNN1GAACHRM3ALDH1A1
SCHEMBL7972494 0.67 MAOB (0.55) VNN1GAACHRM3ALDH1A1
SCHEMBL5091359 0.67 CHRM3 (0.54) VNN1GAAGPR139CHRM3ROCK2
SCHEMBL7233161 0.67 CHRM3 (0.54) VNN1GAAGPR139CHRM3ROCK2
SCHEMBL7983783 0.66 MAOB (0.54) VNN1GAACHRM3ALDH1A1
SCHEMBL5099622 0.66 ROCK2 (0.62) GAAGPR139CHRM3ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015048503-A2 N-ARYLMETHYL SULFONAMIDE NEGATIVE MODULATORS OF NR2A MNEMOSYNE PHARMACEUTICALS, INC. (US) 2015-04-02 WO disclosed