SCHEMBL16619320

SCHEMBL16619320

CC(Nc1c([N+](=O)[O-])cnc2cc(Br)c(CCCC#N)cc12)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.38
PRKDC P78527 3/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
PRKCQ Q04759 2/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16619317 1.00 EGFR (0.38) EGFRPRKDCALDH1A1GAAHTT
SCHEMBL16619177 0.86 EGFR (0.45) EGFRPRKDCALDH1A1PIK3CA
SCHEMBL16619179 0.86 EGFR (0.45) EGFRPRKDCALDH1A1PIK3CA
SCHEMBL16619352 0.86 SIRT5 (0.39) ALDH1A1GAAHTTCRHBPCRHR2
SCHEMBL16619354 0.86 SIRT5 (0.39) ALDH1A1GAAHTTCRHBPCRHR2
SCHEMBL16618793 0.84 ALDH1A1 (0.40) ALDH1A1GAAHTTCRHBPCRHR2
SCHEMBL16618796 0.84 ALDH1A1 (0.40) ALDH1A1GAAHTTCRHBPCRHR2
SCHEMBL16619018 0.83 MAPT (0.43) ALDH1A1TP53
SCHEMBL16619572 0.83 EGFR (0.39) EGFRPRKDCALDH1A1GAAHTT
SCHEMBL16619574 0.83 EGFR (0.39) EGFRPRKDCALDH1A1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049629-A1 IMIDAZOQUINOLINE COMPOUNDS AS BROMODOMAIN INHIBITORS Piramal Enterprises Limited (IN) 2015-04-09 WO disclosed