SCHEMBL16619352

SCHEMBL16619352

CC(Nc1c([N+](=O)[O-])cnc2cc(Br)c(CCC(=O)O)cc12)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 2/20 0.39
ALDH1A1 P00352 5/20 0.39
HTT P42858 3/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 5/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
RECQL P46063 1/20 0.37
PRKCQ Q04759 2/20 0.37
PLK1 P53350 1/20 0.37
TP53 P04637 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16619354 1.00 SIRT5 (0.39) SIRT5ALDH1A1HTTGAAMAPT
SCHEMBL16619018 0.92 MAPT (0.43) ALDH1A1MAPTTP53CYP2C9CYP2C19
SCHEMBL16618796 0.91 ALDH1A1 (0.40) ALDH1A1HTTGAAMAPTNPSR1
SCHEMBL16618793 0.91 ALDH1A1 (0.40) ALDH1A1HTTGAAMAPTNPSR1
SCHEMBL16619487 0.87 EGFR (0.39) PLK1KDM4E
SCHEMBL16619317 0.86 EGFR (0.38) ALDH1A1HTTGAACRHBPCRHR2
SCHEMBL16619320 0.86 EGFR (0.38) ALDH1A1HTTGAACRHBPCRHR2
SCHEMBL16619418 0.84 KDM4E (0.46) ALDH1A1HTTGAAMAPTNPSR1
SCHEMBL16619416 0.84 KDM4E (0.46) ALDH1A1HTTGAAMAPTNPSR1
SCHEMBL16619219 0.83 ALDH1A1 (0.49) ALDH1A1HTTGAAMAPTCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049629-A1 IMIDAZOQUINOLINE COMPOUNDS AS BROMODOMAIN INHIBITORS Piramal Enterprises Limited (IN) 2015-04-09 WO disclosed