SCHEMBL16623477

SCHEMBL16623477

N=C(c1ccc(CN2CCCC2=O)cc1)c1c(Nc2c(F)cccc2F)c(CI)c[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
WDR91 A4D1P6 2/20 0.34
CDC7 O00311 1/20 0.33
PLK4 O00444 1/20 0.33
AURKA O14965 1/20 0.33
MAPK13 O15264 1/20 0.33
PDPK1 O15530 1/20 0.33
DYRK3 O43781 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
ERBB2 P04626 1/20 0.33
NTRK1 P04629 1/20 0.33
PRKCG P05129 1/20 0.33
FYN P06241 1/20 0.33
CSF1R P07333 1/20 0.33
RET P07949 1/20 0.33
IGF1R P08069 1/20 0.33
ROS1 P08922 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849211 0.89 L3MBTL1 (0.38) BDKRB1L3MBTL1WDR91CDC7PLK4
SCHEMBL17849238 0.82 L3MBTL1 (0.38) BDKRB1L3MBTL1WDR91CDC7PLK4
SCHEMBL17849209 0.76 BDKRB1 (0.35) BDKRB1SMN1; SMN2KMT2A
SCHEMBL17849208 0.76 HDAC6 (0.33) HDAC1HDAC6SMN1; SMN2KMT2A
SCHEMBL17849193 0.74 F10 (0.43) PRKAA1RAB9ASMN1; SMN2F10
SCHEMBL17849190 0.74 LTA4H (0.33) NTRK1PARP1RAB9A
SCHEMBL16623476 0.74
SCHEMBL16623450 0.70 NPC1 (0.32)
SCHEMBL16623563 0.69 KMT2A (0.32) KMT2A
SCHEMBL16726665 0.69 ALDH2 (0.33) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed