SCHEMBL17849211

SCHEMBL17849211

N=C(c1ccc(CN2CCCC2=O)cc1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.38
WDR91 A4D1P6 2/20 0.37
HDAC1 Q13547 6/20 0.36
HDAC6 Q9UBN7 3/20 0.36
BDKRB1 P46663 1/20 0.36
RAB9A P51151 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
CDC7 O00311 1/20 0.34
PLK4 O00444 1/20 0.34
AURKA O14965 1/20 0.34
MAPK13 O15264 1/20 0.34
PDPK1 O15530 1/20 0.34
DYRK3 O43781 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PAK4 O96013 1/20 0.34
ERBB2 P04626 1/20 0.34
NTRK1 P04629 1/20 0.34
PRKCG P05129 1/20 0.34
FYN P06241 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16623477 0.89 BDKRB1 (0.36) L3MBTL1WDR91HDAC1HDAC6BDKRB1
SCHEMBL17849208 0.87 HDAC6 (0.33) HDAC1HDAC6ALDH1A1SMN1; SMN2KMT2A
SCHEMBL17849209 0.87 BDKRB1 (0.35) BDKRB1KDM4EALDH1A1SMN1; SMN2MEN1
SCHEMBL17849193 0.85 F10 (0.43) RAB9APRKAA1F10ALDH1A1SMN1; SMN2
SCHEMBL17849190 0.85 LTA4H (0.33) RAB9ANTRK1PARP1ALDH1A1
SCHEMBL17849238 0.85 L3MBTL1 (0.38) L3MBTL1WDR91HDAC1HDAC6BDKRB1
SCHEMBL17849189 0.84 RAB9A (0.45) RAB9AHRH3NTRK1KDM4EALDH1A1
SCHEMBL16623450 0.81 NPC1 (0.32)
SCHEMBL16726665 0.80 ALDH2 (0.33) KMT2A
SCHEMBL16623587 0.79 ROCK1 (0.39) L3MBTL1HDAC1HDAC6RAB9ANTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed