SCHEMBL17849209

SCHEMBL17849209

N=C(c1csc(CN2CCCC2=O)c1)c1c(Nc2c(F)cccc2F)c(Cl)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30
GHSR Q92847 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17849211 0.87 L3MBTL1 (0.38) BDKRB1SMN1; SMN2KDM4EALDH1A1MEN1
SCHEMBL17849200 0.86 CYP2A13 (0.39) SMN1; SMN2ALDH1A1
SCHEMBL18052608 0.82 MEN1 (0.31) MEN1KMT2A
SCHEMBL16623468 0.81 MPO (0.31)
SCHEMBL17849193 0.78 F10 (0.43) SMN1; SMN2ALDH1A1
SCHEMBL17849192 0.77 RIPK1 (0.37) SMN1; SMN2KDM4EKMT2A
SCHEMBL16623477 0.76 BDKRB1 (0.36) BDKRB1SMN1; SMN2KMT2A
SCHEMBL16623544 0.76 MEN1 (0.32) MEN1KMT2A
SCHEMBL17849208 0.76 HDAC6 (0.33) SMN1; SMN2ALDH1A1KMT2A
SCHEMBL17849189 0.74 RAB9A (0.45) SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed
US-9371320-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-21 US disclosed