SCHEMBL16624099

SCHEMBL16624099

COc1ccc2c3c([nH]c2c1)CN(C(C)C)CC3

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.58
ADRA2A P08913 1/20 0.58
ADRA2B P18089 1/20 0.58
ADRA2C P18825 1/20 0.58
NISCH Q9Y2I1 1/20 0.58
CYP2D6 P10635 4/20 0.49
HSD17B10 Q99714 4/20 0.49
KDM4E B2RXH2 4/20 0.49
TSHR P16473 3/20 0.49
MEN1 O00255 2/20 0.49
ALDH1A1 P00352 2/20 0.49
GLA P06280 2/20 0.49
CYP3A4 P08684 2/20 0.49
HPGD P15428 2/20 0.49
CASP1 P29466 2/20 0.49
CASP7 P55210 2/20 0.49
KMT2A Q03164 2/20 0.49
POLB P06746 2/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18034945 0.85 CYP2D6 (0.62) HTR7ADRA2AADRA2BADRA2CNISCH
SCHEMBL17993835 0.82 KDM4E (0.46) KDM4EACHETRPV1BAZ2BCDK4
SCHEMBL17993840 0.82 HTR7 (0.55) HTR7ADRA2AADRA2BADRA2CNISCH
SCHEMBL17993837 0.81 ADRA1A (0.45) KDM4EMEN1KMT2AADRA1ATRPV1
SCHEMBL29564708 0.81 CYP2D6 (0.64) HTR7ADRA2AADRA2BADRA2CNISCH
SCHEMBL25192385 0.81 CYP2D6 (0.64) HTR7ADRA2AADRA2BADRA2CNISCH
SCHEMBL18033535 0.81 KDM4E (0.44) KDM4EMEN1KMT2AMAPTTRPV1
SCHEMBL16624295 0.81 MEN1 (0.45) KDM4EMEN1KMT2AGAAMAPT
SCHEMBL25183522 0.77 HTR7 (0.56) HTR7ADRA2AADRA2BADRA2CNISCH
SCHEMBL16624095 0.77 KIF11 (0.46) KDM4EALDH1A1MAPTTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3053917-A1 T-TYPE CALCIUM CHANNEL BLOCKER Nissan Chemical Industries, Ltd. (JP) 2016-08-10 EP disclosed
WO-2015050212-A1 T-TYPE CALCIUM CHANNEL BLOCKER 日産化学工業株式会社 2015-04-09 WO disclosed