SCHEMBL16627486

SCHEMBL16627486

COC(=O)[C@H](C)n1ccc2cc(Br)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 1/20 0.44
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
MCL1 Q07820 1/20 0.39
NR3C2 P08235 1/20 0.39
KMT2A Q03164 1/20 0.37
FABP4 P15090 2/20 0.37
TP53 P04637 1/20 0.37
KRAS P01116 3/20 0.36
ALDH1A1 P00352 2/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
LMNA P02545 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
FABP3 P05413 1/20 0.36
FABP2 P12104 1/20 0.36
FABP5 Q01469 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16627490 1.00 NTSR1 (0.44) NTSR1HTR2AHTR2CSLC6A2SLC6A4
SCHEMBL16627489 0.86 FPR2 (0.45) NTSR1HTR2AHTR2CSLC6A2SLC6A4
SCHEMBL2000984 0.84 NR3C2 (0.39) SLC6A2SLC6A4NR3C2KMT2ATP53
SCHEMBL2000119 0.84 NR3C2 (0.39) SLC6A2SLC6A4NR3C2KMT2ATP53
SCHEMBL22798848 0.84 NTSR1 (0.50) NTSR1HTR2AHTR2CSLC6A2SLC6A4
SCHEMBL16619844 0.84 NTSR1 (0.50) NTSR1HTR2AHTR2CSLC6A2SLC6A4
SCHEMBL16627458 0.84 NTSR1 (0.50) NTSR1HTR2AHTR2CSLC6A2SLC6A4
SCHEMBL2012022 0.82 HTR2A (0.49) NTSR1HTR2AHTR2CSLC6A2SLC6A4
SCHEMBL2182449 0.79 NR3C2 (0.53) SLC6A2SLC6A4NR3C2KMT2A
SCHEMBL1995408 0.77 ITGB3 (0.41) SLC6A2SLC6A4MCL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049668-A1 NOVEL COMPOUND AS A DIACYLGLYCEROL ACYLTRANSFERASE INHIBITOR GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2015-04-09 WO disclosed