SCHEMBL1663243

SCHEMBL1663243

C#Cc1nc(-c2ccccc2)c(CC=O)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 9/20 0.39
KDM4E B2RXH2 2/20 0.39
POLB P06746 1/20 0.39
CYP1A2 P05177 1/20 0.38
MAPT P10636 5/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ALDH1A1 P00352 4/20 0.38
KMT2A Q03164 4/20 0.37
NPSR1 Q6W5P4 2/20 0.37
TP53 P04637 1/20 0.37
RXFP1 Q9HBX9 2/20 0.36
MEN1 O00255 3/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
PPARG P37231 1/20 0.35
NCOA2 Q15596 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10281014 0.77 PTGDR2 (0.48) PTGDR2KDM4EPOLBCYP1A2MAPT
SCHEMBL28053564 0.67 PTGDR2 (0.34) PTGDR2KDM4EPOLBCYP1A2MAPT
SCHEMBL1664739 0.66 ADORA1 (0.38) KDM4EPOLBMAPTGAASMN1; SMN2
SCHEMBL851867 0.65 SMN1; SMN2 (0.51) PTGDR2KDM4EPOLBMAPTGAA
SCHEMBL19287156 0.65 GAA (0.55) PTGDR2KDM4EMAPTGAASMN1; SMN2
SCHEMBL3995474 0.60 CKS1B (0.45) KMT2ATP53MEN1LMNATDP1
SCHEMBL3993059 0.60 S1PR3 (0.50) KDM4EHSD17B10ALDH1A1KMT2AMEN1
SCHEMBL2544178 0.59 PTPN1 (0.47)
SCHEMBL5746080 0.59 MAPT (0.49) KDM4ECYP1A2MAPTGAASMN1; SMN2
SCHEMBL5147356 0.59 BCAT2 (0.43) PTGDR2ALDH1A1KMT2ATP53RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2490541-A1 2-SUBSTITUTED-ETHYNYLTHIAZOLE DERIVATIVES AND USES OF SAME H. Lundbeck A/S (DK) 2012-08-29 EP disclosed
WO-2011050063-A1 2-SUBSTITUTED-ETHYNYLTHIAZOLE DERIVATIVES AND USES OF SAME H. LUNDBECK A/S (DK) 2011-04-28 WO disclosed