SCHEMBL16634671

SCHEMBL16634671

O=C(O)c1ccc(-n2c(=O)n(C(=O)c3c(Cl)cccc3Cl)c3cc(NCC4CCC4)ccc32)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.39
RORC P51449 14/20 0.37
CYP3A4 P08684 2/20 0.34
CRHR1 P34998 1/20 0.34
LDHA P00338 1/20 0.33
LDHB P07195 1/20 0.33
RARG P13631 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK10 P53779 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634673 0.79 RORC (0.40) RORCCYP3A4RARGCYP1A2CYP2C9
SCHEMBL16634649 0.78 RORC (0.43) RORCCYP3A4RARGCYP1A2CYP2C9
SCHEMBL16634554 0.76 RORC (0.55) RORCCYP3A4RARGCYP1A2CYP2C9
SCHEMBL16634751 0.74 RORC (0.42) RORCCYP3A4RARGCYP1A2CYP2C9
SCHEMBL16634779 0.73 RORC (0.53) RORCCYP3A4RARGCYP1A2CYP2C9
SCHEMBL16634532 0.73 AURKA (0.41) LTA4H
SCHEMBL16634721 0.70 RAB9A (0.45) RORC
SCHEMBL16634636 0.68 RORC (0.56) RORCCYP3A4CYP2C9CYP2C19
SCHEMBL16634830 0.67 RORC (0.43) RORCCYP3A4RARGCYP1A2CYP2C9
SCHEMBL16634665 0.67 ALDH1A1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO claimed
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed