SCHEMBL16637128

SCHEMBL16637128

N#Cc1ccc(N2CC3(CC3)CC(Cl)(Cl)C2=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.40
ELANE P08246 1/20 0.39
POLB P06746 1/20 0.39
NSD2 O96028 1/20 0.39
OPRM1 P35372 2/20 0.39
OPRL1 P41146 2/20 0.39
PGR P06401 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
RAB9A P51151 1/20 0.37
METAP2 P50579 1/20 0.35
KCNJ1 P48048 1/20 0.35
CYP2D6 P10635 2/20 0.34
ACACA Q13085 1/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16324730 0.81 RAB9A (0.40) POLBL3MBTL1SMN1; SMN2RAB9A
SCHEMBL16637430 0.79 OPRM1 (0.44) NSD2OPRM1OPRL1L3MBTL1SMN1; SMN2
SCHEMBL16637299 0.75 POLB (0.45) CYP11B2ELANEPOLBNSD2OPRM1
SCHEMBL16430910 0.69 ACACA (0.48) CYP11B2ELANEPOLBOPRM1OPRL1
SCHEMBL21753280 0.64 ACACA (0.56) POLBKCNJ1CYP2D6ACACATSHR
SCHEMBL6740517 0.64 POLB (0.46) CYP11B2ELANEPOLBOPRM1OPRL1
SCHEMBL21764939 0.64 USP2 (0.43) ELANEPOLBOPRM1OPRL1PGR
SCHEMBL7422542 0.63 POLB (0.49) CYP11B2ELANEPOLB
Hydrochloric Acid SCHEMBL21753301 0.63 USP2 (0.42) ELANEPOLBOPRM1OPRL1PGR
SCHEMBL23299517 0.63 GRM2 (0.43) CYP11B2ELANEPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed