SCHEMBL16637430

SCHEMBL16637430

N#Cc1ccc(N2CC3(CC3)CC(Cl)(Cl)C2=O)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.44
OPRL1 P41146 3/20 0.44
ACACA Q13085 1/20 0.40
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
CRHR1 P34998 1/20 0.35
NSD2 O96028 1/20 0.34
PARP1 P09874 4/20 0.33
PARP2 Q9UGN5 2/20 0.33
TRPV4 Q9HBA0 1/20 0.33
ALDH1A1 P00352 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
AOC3 Q16853 1/20 0.32
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CASP3 P42574 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
TNK1 Q13470 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637128 0.79 CYP11B2 (0.40) OPRM1OPRL1ACACANSD2SMN1; SMN2
SCHEMBL16637361 0.79 OPRM1 (0.47) OPRM1OPRL1ACACAADRA1DADRA1A
SCHEMBL11543022 0.66 KDM4E (0.37) OPRM1OPRL1ADRA1DADRA1AADRA1B
SCHEMBL11539917 0.65 KDM4E (0.38) OPRM1OPRL1ADRA1DADRA1AADRA1B
SCHEMBL249165 0.64 PDE3B (0.43) ADRA1DADRA1AADRA1BALDH1A1AOC3
SCHEMBL16324730 0.64 RAB9A (0.40) SMN1; SMN2L3MBTL1
Hydrochloric Acid SCHEMBL6361748 0.63 FPR2 (0.43) OPRM1OPRL1ADRA1DADRA1AADRA1B
SCHEMBL31686991 0.62 SLC6A9 (0.45) ADRA1DADRA1AADRA1BALDH1A1AOC3
SCHEMBL15212468 0.62 OPRM1 (0.41) OPRM1OPRL1ADRA1DADRA1AADRA1B
SCHEMBL251355 0.62 SLC6A9 (0.45) OPRM1OPRL1ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed