SCHEMBL16637238

SCHEMBL16637238

CN(C)C(=O)c1ccc(N2CC3(CC3)CC(Cl)(Cl)C2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.42
OPRM1 P35372 3/20 0.39
OPRL1 P41146 3/20 0.39
GAA P10253 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
RAB9A P51151 1/20 0.36
HPGD P15428 2/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
GRIA2 P42262 1/20 0.33
MAPT P10636 1/20 0.33
OTUD7B Q6GQQ9 3/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
HDAC1 Q13547 3/20 0.32
HDAC8 Q9BY41 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637329 0.77 OPRM1 (0.41) L3MBTL1OPRM1OPRL1GAASMN1; SMN2
SCHEMBL1004649 0.64 ALDH1A1 (0.73) SMN1; SMN2HPGDALDH1A1CYP1A2CYP2D6
SCHEMBL9595456 0.64 KMT2A (0.66) GAASMN1; SMN2RAB9AHPGDALDH1A1
SCHEMBL9431536 0.62 SMN1; SMN2 (0.55) L3MBTL1GAASMN1; SMN2RAB9AALDH1A1
SCHEMBL5639628 0.61 OPRM1 (0.39) L3MBTL1OPRM1OPRL1GAASMN1; SMN2
SCHEMBL487487 0.61 HPGD (0.61) SMN1; SMN2HPGDALDH1A1MAPT
SCHEMBL15387038 0.61 HPGD (0.52) GAASMN1; SMN2HPGDALDH1A1CYP1A2
SCHEMBL28513427 0.60 GAA (0.47) L3MBTL1GAASMN1; SMN2RAB9AHPGD
SCHEMBL10405466 0.60 ALDH1A1 (0.63) L3MBTL1SMN1; SMN2RAB9AHPGDALDH1A1
SCHEMBL31702358 0.59 GFER (0.43) OPRM1OPRL1GAASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed