SCHEMBL16637329

SCHEMBL16637329

CN(C)C(=O)c1ccc(N2CC3(CCC2=O)CC3)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.41
OPRL1 P41146 3/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 4/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 1/20 0.37
GRIA2 P42262 1/20 0.37
ITGB3 P05106 4/20 0.37
ITGA2B P08514 4/20 0.37
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16644311 0.82 ALDH1A1 (0.59) ALDH1A1HPGDCYP1A2CYP2D6ITGB3
SCHEMBL16637238 0.77 L3MBTL1 (0.42) OPRM1OPRL1ALDH1A1HPGDL3MBTL1
SCHEMBL16361765 0.77 TP53 (0.44) OPRM1OPRL1SMN1; SMN2GAAMAPT
SCHEMBL16637490 0.76 HPGD (0.67) ALDH1A1HPGDSMN1; SMN2GAA
SCHEMBL16361938 0.74 SLC6A2 (0.38) ALDH1A1SMN1; SMN2ITGB3ITGA2BRAB9A
SCHEMBL16637299 0.71 POLB (0.45) OPRM1OPRL1SMN1; SMN2CYP2D6
SCHEMBL25315488 0.67 ACACB (0.46) SMN1; SMN2ITGB3ITGA2BMAPT
SCHEMBL1004649 0.67 ALDH1A1 (0.73) ALDH1A1HPGDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL13664713 0.66 SLC6A2 (0.57) OPRM1OPRL1ALDH1A1L3MBTL1ITGB3
SCHEMBL738643 0.65 TSHR (0.54) ALDH1A1HPGDSMN1; SMN2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed
WO-2015051713-A1 4,5-DIHYDRO-PYRAZOLO[3,4-C]PYRIDIN-2-ONE SPIRO DERIVATIVE, PREPARATION METHOD AND USE THEREOF 四川海思科制药有限公司 2015-04-16 WO disclosed