SCHEMBL16664374

SCHEMBL16664374

O=C(O)[C@H](CNc1cccc(OC(F)(F)F)c1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 1/20 0.46
CASR P41180 1/20 0.44
EPHX2 P34913 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.43
P2RX1 P51575 1/20 0.43
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2487961 0.78 MMP12 (0.48) GPR139CASREPHX2ALDH1A1GAA
SCHEMBL13240798 0.78 MMP12 (0.48) GPR139CASREPHX2ALDH1A1GAA
SCHEMBL13285509 0.78 CYP2C19 (0.50) ALDH1A1MAPTHTT
SCHEMBL3611216 0.77 ALDH1A1 (0.50) EPHX2ALDH1A1GAAMAPTHPGD
Hydrochloric Acid SCHEMBL2487924 0.77 MMP12 (0.47) GPR139CASREPHX2ALDH1A1GAA
SCHEMBL6748392 0.76 CETP (0.54) ALDH1A1GAAMAPTHPGDALOX15
SCHEMBL8351967 0.76 ICMT (0.44) GPR139EPHX2ALDH1A1GAAMAPT
SCHEMBL16028565 0.75 AKR1C3 (0.51) GPR139TRPM8
SCHEMBL16664416 0.75 MEN1 (0.46) ALDH1A1MAPTHPGDTSHRHTT
SCHEMBL13282525 0.73 CNR2 (0.48) MAPTHPGDHDAC4HDAC7HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376489-B1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF CHIESI FARMA SPA (IT) 2015-04-22 EP disclosed