SCHEMBL16664911

SCHEMBL16664911

CCCNc1cc(-c2cnc(OCC(F)(F)F)nc2)ncn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 8/20 0.43
TSHR P16473 5/20 0.43
CYP1A2 P05177 5/20 0.43
CYP2C19 P33261 5/20 0.43
CYP3A4 P08684 3/20 0.43
KDM4E B2RXH2 1/20 0.43
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
USP2 O75604 2/20 0.38
CYP2D6 P10635 2/20 0.38
HIF1A Q16665 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
TRPV3 Q8NET8 1/20 0.38
BRAF P15056 1/20 0.37
KDR P35968 1/20 0.37
MAPK14 Q16539 1/20 0.37
TNNI3K Q59H18 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664909 0.85 CYP1A2 (0.43) FAAHTSHRCYP1A2CYP2C19CYP3A4
SCHEMBL16664949 0.76 FLT3 (0.39) FAAHTSHRCYP1A2CYP2C19CYP3A4
SCHEMBL16664979 0.76 FAAH (0.39) FAAHTSHRCYP1A2CYP2C19CYP3A4
SCHEMBL16665010 0.76 FAAH (0.41) FAAHCYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL18627048 0.74 ABL1 (0.44) FAAHTSHRCYP1A2CYP2C19CYP3A4
SCHEMBL15473168 0.74 FAAH (0.43) FAAHTSHRCYP1A2CYP2C19CYP3A4
SCHEMBL19819911 0.73 HPGDS (0.37) TSHRCYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL16664919 0.72 PIK3CA (0.44) FAAHCYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL16664969 0.72 KDM4E (0.47) FAAHCYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL15473146 0.72 CYP1A2 (0.36) FAAHTSHRCYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed