SCHEMBL16664960

SCHEMBL16664960

CNC(=O)c1ccc(CS)c(OC)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.49
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
HPGD P15428 2/20 0.48
ALDH1A1 P00352 1/20 0.48
CCNC P24863 1/20 0.44
CDK8 P49336 1/20 0.44
HDAC8 Q9BY41 2/20 0.43
PYGL P06737 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
MAPK1 P28482 1/20 0.42
TSHR P16473 2/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15356444 0.87 PLK1 (0.51) PLK1SLC6A2SLC6A4SLC6A3HPGD
SCHEMBL9364255 0.84 MAPT (0.57) HPGDALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL22838519 0.83 PLK1 (0.53) PLK1SLC6A2SLC6A4SLC6A3HPGD
SCHEMBL9428447 0.82 CA12 (0.62) ALDH1A1LMNAMAPK1TSHRCYP1A2
SCHEMBL4151619 0.80 CYP1A2 (0.66) PLK1HPGDALDH1A1CCNCCDK8
SCHEMBL15342989 0.79 PLK1 (0.53) PLK1SLC6A2SLC6A4SLC6A3HPGD
SCHEMBL17758615 0.78 SLC6A2 (0.56) PLK1SLC6A2SLC6A4SLC6A3HPGD
SCHEMBL9103250 0.77 TAS1R3 (0.56) PLK1SLC6A2SLC6A4SLC6A3HPGD
SCHEMBL5758000 0.77 MEN1 (0.68) PLK1HPGDALDH1A1MAPTALOX15
SCHEMBL72600 0.76 PLK1 (0.53) PLK1SLC6A2SLC6A4SLC6A3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed