SCHEMBL16664967

SCHEMBL16664967

CCCNc1cc(-c2ccnc(OC)c2)ncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 16/20 0.45
CYP2C19 P33261 16/20 0.45
CLK4 Q9HAZ1 15/20 0.45
CYP3A4 P08684 15/20 0.45
CYP2D6 P10635 14/20 0.45
TSHR P16473 11/20 0.45
MAPK1 P28482 6/20 0.45
HSD17B10 Q99714 7/20 0.44
TP53 P04637 4/20 0.44
HIF1A Q16665 3/20 0.44
ALOX15 P16050 5/20 0.43
LMNA P02545 5/20 0.43
ALDH1A1 P00352 10/20 0.42
USP2 O75604 5/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CDC7 O00311 1/20 0.42
ROCK2 O75116 1/20 0.42
MAP4K4 O95819 1/20 0.42
PIM1 P11309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664939 0.90 CLK4 (0.42) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL16660240 0.84 FAAH (0.48) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL16664988 0.82 CLK4 (0.44) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL12963406 0.80 DNM2 (0.43) CYP1A2CYP2C19CLK4TSHRTP53
SCHEMBL18627048 0.78 ABL1 (0.44) CYP1A2CYP2C19CLK4CYP3A4TSHR
SCHEMBL12907692 0.78 ABL1 (0.45) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL18902711 0.76 CYP1A2 (0.53) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL19905341 0.73 ASIC3 (0.50) MEN1KMT2AGSK3BMAPTPIK3CA
SCHEMBL16664965 0.73 PIK3CA (0.40) CYP1A2CYP2C19CLK4CYP3A4CYP2D6
SCHEMBL16664987 0.73 CYP1A2 (0.46) CYP1A2CYP2C19CLK4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed