SCHEMBL16664987

SCHEMBL16664987

CCCNc1cc(-c2cnc(OC)c(OC)c2)ncn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 17/20 0.46
CYP2D6 P10635 16/20 0.46
CYP2C19 P33261 15/20 0.46
CYP3A4 P08684 14/20 0.46
CLK4 Q9HAZ1 14/20 0.46
TSHR P16473 14/20 0.46
HSD17B10 Q99714 9/20 0.46
ALDH1A1 P00352 9/20 0.43
TP53 P04637 6/20 0.43
MAPK1 P28482 6/20 0.43
LMNA P02545 5/20 0.43
HIF1A Q16665 5/20 0.43
CYP2C9 P11712 2/20 0.43
ALOX15 P16050 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
USP2 O75604 3/20 0.41
FYN P06241 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664990 0.86 MAPT (0.45) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16664971 0.83 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL19355497 0.74 CYP1A2 (0.41) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16664927 0.74 FAAH (0.38) CYP1A2CYP2C19CYP3A4TSHRHSD17B10
SCHEMBL16664979 0.73 FAAH (0.39) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16665010 0.73 FAAH (0.41) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16664967 0.73 CYP1A2 (0.45) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16664919 0.72 PIK3CA (0.44) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16664909 0.72 CYP1A2 (0.43) CYP1A2CYP2D6CYP2C19CYP3A4CLK4
SCHEMBL16664969 0.72 KDM4E (0.47) CYP1A2CYP2D6CYP2C19CYP3A4CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed