SCHEMBL16664971

SCHEMBL16664971

CCCNc1cc(-c2cnc(C#N)c(OC)c2)ncn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 16/20 0.46
CLK4 Q9HAZ1 15/20 0.46
CYP3A4 P08684 14/20 0.46
CYP2C19 P33261 14/20 0.46
TSHR P16473 12/20 0.46
ALDH1A1 P00352 10/20 0.46
MAPK1 P28482 6/20 0.46
CYP2D6 P10635 13/20 0.43
USP2 O75604 5/20 0.43
HSD17B10 Q99714 7/20 0.41
LMNA P02545 5/20 0.40
TP53 P04637 5/20 0.40
HIF1A Q16665 5/20 0.40
CYP2C9 P11712 2/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
ALOX15 P16050 1/20 0.39
FYN P06241 2/20 0.38
HPGD P15428 1/20 0.38
GLA P06280 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15343321 0.85 CYP1A2 (0.45) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL16664987 0.83 CYP1A2 (0.46) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL16664934 0.75 CYP1A2 (0.39) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL16664990 0.75 MAPT (0.45) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL19905177 0.73 CYP1A2 (0.42) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL16664979 0.70 FAAH (0.39) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL16665010 0.70 FAAH (0.41) CYP1A2CLK4CYP3A4CYP2C19ALDH1A1
SCHEMBL16664967 0.69 CYP1A2 (0.45) CYP1A2CLK4CYP3A4CYP2C19TSHR
SCHEMBL16664919 0.69 PIK3CA (0.44) CYP1A2CLK4CYP3A4CYP2C19ALDH1A1
SCHEMBL16664969 0.69 KDM4E (0.47) CYP1A2CLK4CYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed