SCHEMBL16668583

SCHEMBL16668583

Brc1ccc(OBOc2ccc(Br)c3ccccc23)c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.47
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GPR84 Q9NQS5 1/20 0.39
RXFP1 Q9HBX9 1/20 0.35
HTR6 P50406 1/20 0.34
AAK1 Q2M2I8 1/20 0.33
IDO1 P14902 1/20 0.32
NQO2 P16083 1/20 0.32
EP300 Q09472 1/20 0.31
KAT8 Q9H7Z6 1/20 0.31
PRNP P04156 1/20 0.31
CYP1A2 P05177 1/20 0.31
PARP1 P09874 1/20 0.31
NQO1 P15559 1/20 0.30
EPHX1 P07099 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15449549 0.83 PKM (0.49) PKMLMNAL3MBTL1GPR84RXFP1
SCHEMBL11068046 0.79 PKM (0.52) PKMLMNAL3MBTL1GPR84RXFP1
SCHEMBL30719614 0.76 IDO1 (0.57) PKMLMNAL3MBTL1IDO1NQO2
SCHEMBL1891196 0.76 IDO1 (0.57) PKMLMNAL3MBTL1IDO1NQO2
SCHEMBL30710586 0.75 RXFP1 (0.48) PKMLMNAL3MBTL1RXFP1HTR6
SCHEMBL198796 0.75 RXFP1 (0.48) PKMLMNAL3MBTL1RXFP1HTR6
SCHEMBL29429114 0.75 RXFP1 (0.48) PKMLMNAL3MBTL1RXFP1HTR6
SCHEMBL15901381 0.74 GPR84 (0.39) GPR84IDO1EP300KAT8NQO1
SCHEMBL904667 0.74 CYP1A2 (0.56) LMNAL3MBTL1IDO1EP300KAT8
SCHEMBL7527797 0.74 IDO1 (0.55) PKMLMNAL3MBTL1IDO1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127261-A1 COMPOUND AND PREPARATION METHOD THEREOF AND APPLICATION THEREOF IN PREPARATION OF THERAPEUTIC ANTI-CANCER DRUG 天津济坤医药科技有限公司 2022-06-23 WO disclosed
CN-112574216-B Compound, preparation method thereof and application thereof in preparing anti-cancer drugs 天津济坤医药科技有限公司 2022-03-08 CN disclosed
CN-112574216-A Compound, preparation method thereof and application thereof in preparing anti-cancer drugs 天津济坤医药科技有限公司 2021-03-30 CN disclosed
US-9601699-B2 Chrysene-based compound and organic light-emitting device including the same SAMSUNG DISPLAY CO., LTD. (KR) 2017-03-21 US disclosed
US-20150115232-A1 CHRYSENE-BASED COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG DISPLAY CO., LTD. (KR) 2015-04-30 US disclosed