SCHEMBL16684544

SCHEMBL16684544

O=S(=O)(OC1=C(COCc2ccccc2)CCCC1)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
CA2 P00918 2/20 0.38
DRD2 P14416 2/20 0.35
DRD1 P21728 2/20 0.35
DRD4 P21917 2/20 0.35
DRD5 P21918 2/20 0.35
DRD3 P35462 2/20 0.35
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
LTA4H P09960 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
RORC P51449 3/20 0.33
NR1I2 O75469 1/20 0.33
PTPRZ1 P23471 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21138206 0.75 ALDH1A1 (0.43) TSHRCA2CA1CA9LMNA
SCHEMBL5668749 0.75
SCHEMBL12354193 0.73 DRD2 (0.34) DRD2DRD1DRD4DRD5DRD3
SCHEMBL17395579 0.73
SCHEMBL4160550 0.71 PTGS2 (0.41) CA2DRD2DRD1DRD4DRD5
SCHEMBL6163354 0.70 DRD2 (0.34) DRD2DRD1DRD4DRD5DRD3
SCHEMBL19141072 0.70
SCHEMBL8388405 0.69 RXRA (0.30)
SCHEMBL17314725 0.68 PTGS2 (0.38) DRD2DRD1DRD4DRD5DRD3
SCHEMBL8499207 0.67 CA12 (0.58) CA2CA1CA9LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116640094-A Compounds as PRMT1 inhibitors and uses thereof 南京圣和药业股份有限公司 2023-08-25 CN disclosed
EP-3063143-A1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS Novartis AG (CH) 2016-09-07 EP disclosed
WO-2015066188-A1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS AG (CH) 2015-05-07 WO disclosed