SCHEMBL1668599

SCHEMBL1668599

CN1CC(c2ccccc2)(c2cc(CCCOCCC(=O)O)ccc2O)C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.38
CHRM5 P08912 3/20 0.37
CHRM1 P11229 3/20 0.37
CHRM3 P20309 3/20 0.37
FFAR1 O14842 1/20 0.36
S1PR1 P21453 5/20 0.36
S1PR5 Q9H228 3/20 0.36
S1PR3 Q99500 2/20 0.36
ALOX5 P09917 1/20 0.35
DRD4 P21917 1/20 0.35
OPRM1 P35372 1/20 0.35
CYP1A2 P05177 1/20 0.35
SLC6A4 P31645 1/20 0.34
APP P05067 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800404 0.94 CHRM5 (0.40) RXRACHRM5CHRM1CHRM3FFAR1
SCHEMBL1668720 0.91 CHRM5 (0.43) RXRACHRM5CHRM1CHRM3S1PR1
SCHEMBL1668322 0.85 S1PR1 (0.40) CHRM5CHRM1CHRM3S1PR1S1PR5
SCHEMBL12801191 0.84 CHRM5 (0.46) RXRACHRM5CHRM1CHRM3DRD4
SCHEMBL1668419 0.84 RXRA (0.38) RXRACHRM5CHRM1CHRM3S1PR1
SCHEMBL1668486 0.83 SMN1; SMN2 (0.43) RXRACHRM5CHRM1CHRM3FFAR1
SCHEMBL1670818 0.81 FFAR4 (0.37) RXRACHRM5CHRM1CHRM3OPRM1
SCHEMBL1668622 0.81 OPRD1 (0.36) OPRM1APPFFAR4
SCHEMBL1668421 0.81 FFAR4 (0.37) RXRACHRM5CHRM1CHRM3OPRM1
SCHEMBL12800754 0.80 OPRM1 (0.33) CHRM5CHRM1CHRM3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed