SCHEMBL1669065

SCHEMBL1669065

O=c1[nH]cnc2ccc(N3CCN4CCCCCCCCCCCCCCCCCCCCCC3CC4)cc12

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 12/20 0.60
IP6K3 Q96PC2 4/20 0.58
IP6K2 Q9UHH9 1/20 0.54
CHRNA7 P36544 2/20 0.46
PARP1 P09874 4/20 0.40
CHEK1 O14757 1/20 0.40
PIM1 P11309 1/20 0.40
AKT1 P31749 1/20 0.40
FLT3 P36888 1/20 0.40
PIM3 Q86V86 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6886644 0.93 IP6K1 (0.59) IP6K1IP6K3IP6K2CHRNA7PARP1
SCHEMBL1672235 0.80 CHRNA7 (0.45) IP6K1CHRNA7
SCHEMBL1669111 0.79 HPGD (0.46) CHRNA7PARP1
SCHEMBL8871369 0.76 IP6K1 (1.00) IP6K1IP6K3IP6K2
SCHEMBL1670541 0.76 CHRNA7 (0.44) CHRNA7PARP1
SCHEMBL8976326 0.74 IP6K1 (1.00) IP6K1IP6K3IP6K2CHEK1PIM1
SCHEMBL1669269 0.74 TNKS (0.44) CHRNA7PARP1
SCHEMBL6886724 0.74 ACVR1 (0.49) CHRNA7
SCHEMBL6886458 0.71 CHRNA7 (0.50) IP6K1CHRNA7
SCHEMBL6888091 0.70 TNKS (0.51) CHRNA7PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488520-A1 CONDENSED AZINE - DERIVATIVES FOR THE TREATMENT OF DISEASES RELATED TO THE ACETYLCHOLINE RECEPTOR MSD Oss B.V. (NL) 2012-08-22 EP disclosed
WO-2011045258-A1 CONDENSED AZINE - DERIVATIVES FOR THE TREATMENT OF DISEASES RELATED TO THE ACETYLCHOLINE RECEPTOR N.V. ORGANON (NL) 2011-04-21 WO disclosed