SCHEMBL1670381

SCHEMBL1670381

COc1ccc(-c2cn(C)c(C#N)c2I)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GRM2 Q14416 1/20 0.39
ALDH1A1 P00352 5/20 0.38
MAPT P10636 4/20 0.38
KDM4E B2RXH2 4/20 0.38
NPSR1 Q6W5P4 3/20 0.38
RXFP1 Q9HBX9 2/20 0.38
HPGD P15428 2/20 0.38
KMT2A Q03164 7/20 0.38
MEN1 O00255 6/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
LMNA P02545 1/20 0.38
CYP2C9 P11712 1/20 0.38
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670787 0.82 MAPKAPK2 (0.47) MAPKAPK2GABRA1GABRG2GABRB3GABRA3
SCHEMBL28350054 0.76 GRM2 (0.47) MAPKAPK2GABRA1GABRG2GABRB3GABRA3
SCHEMBL12800377 0.76 MAPT (0.44) MAPKAPK2ALDH1A1MAPTKMT2AMEN1
SCHEMBL1671716 0.71 GRIA2 (0.41) ALDH1A1MAPTKDM4ENPSR1RXFP1
SCHEMBL7574828 0.68 KMT2A (0.55) GRM2ALDH1A1MAPTKDM4ENPSR1
SCHEMBL1670712 0.67 PGR (0.44) ALDH1A1MAPTKDM4EHPGDKMT2A
SCHEMBL1185054 0.67 ALDH1A1 (0.47) MAPKAPK2ALDH1A1MAPTKDM4ENPSR1
SCHEMBL12800389 0.66 MAPT (0.44) MAPKAPK2ALDH1A1MAPTKMT2AMEN1
SCHEMBL29663328 0.66 PGR (0.50) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL12670739 0.65 PRKAB2 (0.51) GABRA1GABRG2GABRB3GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed