SCHEMBL1670835

SCHEMBL1670835

CN1CCC(c2ccccc2)(c2cc(C(=O)NCCOCCC(=O)O)ccc2O)CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
NAMPT P43490 2/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HTT P42858 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
CA2 P00918 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
P2RX7 Q99572 1/20 0.37
ADRA1A P35348 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1668840 0.94 NAMPT (0.42) OPRM1NAMPTCA2LMNATP53
Trifluoroacetic Acid SCHEMBL1670826 0.82 ITGB3 (0.41) OPRM1SMN1; SMN2NPC1RAB9AHTT
SCHEMBL12801191 0.81 CHRM5 (0.46) OPRM1OPRD1OPRK1ADRA1ACHRM5
SCHEMBL12801259 0.81 OPRM1 (0.42) OPRM1SMN1; SMN2NPC1RAB9AHTT
SCHEMBL12800770 0.81 OPRD1 (0.42) OPRM1SMN1; SMN2NAMPTHTTHDAC1
SCHEMBL1668720 0.80 CHRM5 (0.43) OPRM1OPRD1OPRK1ADRA1ACHRM5
Trifluoroacetic Acid SCHEMBL1670822 0.78 ITGB3 (0.42) NAMPTHDAC1CA2TP53MAPT
SCHEMBL12801195 0.76 KDM4E (0.42) NAMPTHDAC1OPRD1OPRK1
SCHEMBL12801253 0.76 NAMPT (0.37) OPRM1NAMPTLMNATP53MAPT
SCHEMBL1670831 0.74 SMN1; SMN2 (0.36) OPRM1SMN1; SMN2NPC1RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed