SCHEMBL16712293

SCHEMBL16712293

COc1c(Cl)ccc(-c2nc(O)c(Br)c(C(=O)O)n2)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEP1B Q16820 1/20 0.38
KMO O15229 2/20 0.37
TPMT P51580 2/20 0.36
ACLY P53396 5/20 0.35
TSHR P16473 1/20 0.33
TAS1R3 Q7RTX0 2/20 0.33
TAS1R1 Q7RTX1 2/20 0.33
TAS1R2 Q8TE23 1/20 0.33
PRKAB2 O43741 2/20 0.32
PRKAG1 P54619 2/20 0.32
PRKAA2 P54646 2/20 0.32
PRKAA1 Q13131 2/20 0.32
PRKAG3 Q9UGI9 2/20 0.32
PRKAG2 Q9UGJ0 2/20 0.32
PRKAB1 Q9Y478 2/20 0.32
CDK9 P50750 1/20 0.32
DYRK1A Q13627 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1115150 0.91 MEP1B (0.39) ALDH1A1HSD17B10KDM4EMEP1BACLY
SCHEMBL16712267 0.90 ALDH1A1 (0.43) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL119198 0.89 ALDH1A1 (0.42) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL1223251 0.88 ALDH1A1 (0.41) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL16712268 0.84 ALDH1A1 (0.38) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL119850 0.82 ALDH1A1 (0.43) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL13075707 0.81 ALDH1A1 (0.42) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL1397100 0.81 ALDH1A1 (0.42) ALDH1A1HSD17B10KDM4EMEP1BKMO
SCHEMBL1115268 0.81 TAS1R3 (0.39) ALDH1A1HSD17B10KDM4EMEP1BTPMT
SCHEMBL16712292 0.81 MEP1B (0.38) ALDH1A1HSD17B10KDM4EMEP1BTAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279178-B1 2-(substituted phenyl)-6-hydroxy- or alkoxy-5-substituted-4-pyrimidinecarboxylates and their use as herbicides DOW AGROSCIENCES LLC (US) 2015-05-20 EP claimed