Embusartan

Embusartan

SCHEMBL167147

CCCCc1cc(C(=O)OC)cc(=O)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1F

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 3/20 0.41
AGTR1 P30556 3/20 0.39
AGTR2 P50052 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Embusartan SCHEMBL29409583 1.00 BDKRB1 (0.41) BDKRB1AGTR1AGTR2
Embusartan SCHEMBL5534640 0.95 BDKRB1 (0.38) BDKRB1AGTR1AGTR2
Embusartan SCHEMBL5537210 0.95 BDKRB1 (0.38) BDKRB1AGTR1AGTR2
SCHEMBL5814612 0.91 AGTR1 (0.43) AGTR1AGTR2
SCHEMBL8013981 0.91 AGTR1 (0.39) AGTR1AGTR2
SCHEMBL8009750 0.91
SCHEMBL8007180 0.90
SCHEMBL8433566 0.90
SCHEMBL9412776 0.90 BDKRB1 (0.43) BDKRB1AGTR1AGTR2
Embusartan SCHEMBL5537214 0.90

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1731 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250082608-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2025-03-13 US claimed
EP-4448096-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE Singapore Health Services Pte. Ltd. (SG) 2024-10-23 EP claimed
US-12064429-B2 Substituted 5-fluoro-1H-pyrazolopyridines and their use ADVERIO PHARMA GMBH (DE) 2024-08-20 US claimed
US-12016835-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2024-06-25 US claimed
US-20240173302-A1 TREATMENT OF INFLAMMATORY DISEASES DIMERIX BIOSCIENCE PTY LTD. (AU) 2024-05-30 US claimed
EP-4313024-A1 TREATMENT OF INFLAMMATORY DISEASES Dimerix Bioscience Pty Ltd (AU) 2024-02-07 EP claimed
US-11851443-B2 Neprilysin inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-12-26 US claimed
US-20230285340-A1 NEPRILYSIN INHIBITORS THERAVANCE BIOPHARMA R&D IP LLC (US) 2023-09-14 US claimed
US-11718591-B2 Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2- methylpentanoic acid and uses thereof THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-08-08 US claimed
WO-2023111196-A1 TREATMENT AND PREVENTION OF GLOMERULAR DISEASE SINGAPORE HEALTH SERVICES PTE. LTD. (SG) 2023-06-22 WO claimed
US-20050288272-A1 Pharmaceutical compositions comprising NEP-inhibitors, inhibitors of the endogenous endothelin producing system and AT1 receptor antagonists SOLVAY PHARMACEUTICALS GMBH (DE) 2005-12-29 US claimed
EP-1545540-A2 COMBINATION THERAPY USING A DUAL PPAR ALPHA/GAMMA AGONIST AND AN ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST Merck & Co., Inc. (US) 2005-06-29 EP claimed
WO-2005023182-A2 NITROSATED AND NITROSYLATED CARDIOVASCULAR COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2005-03-17 WO claimed
WO-2004080488-A2 COMBINED PREPARATIONS OF ACETYL SALICYLIC ACID WITH AN HMG-COA REDUCTASE INHIBITOR BAYER HEALTHCARE AG (DE) 2004-09-23 WO claimed
WO-2004017896-A2 COMBINATION THERAPY USING A DUAL PPAR ALPHA/GAMMA AGONIST AND AN ANGIOTENSIN II TYPE I RECEPTOR ANTAGONIST MERCK & CO., INC. (US) 2004-03-04 WO claimed
EP-1258258-A1 Implantable device comprising a stent and angiotensin II receptor antagonists TERUMO KABUSHIKI KAISHA (JP) 2002-11-20 EP claimed
US-20020168393-A1 Implantable medical material and implantable medical device TERUMO KABUSHIKI KAISHA (JP) 2002-11-14 US claimed
WO-2000037075-A1 COMBINATION OF AN AT1 ANGIOTENSIN II RECEPTOR ANTAGONIST AND AN IMMUNOSUPPRESSANT SANOFI-SYNTHELABO (FR) 2000-06-29 WO claimed
EP-0594019-B1 1-Biphenylmethyl-pyridone derivatives, their preparation and their use as angiotensin II antagonistes BAYER AG (DE) 2000-02-23 EP claimed
US-5863930-A ATHEROSCLEROSIS TREATMENT FORMED BY REACTION OF PYRIDONES WITH BIPHENYLMETHYL HALOGEN BAYER AKTIENGESELLSCHAFT (DE) 1999-01-26 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285340-A1 NEPRILYSIN INHIBITORS MME, REN, ACE BDKRB1 41/4885AGTR1 5/4885AGTR2 11/4885
US-12064429-B2 Substituted 5-fluoro-1H-pyrazolopyridines and their use PFKP, PON1, FABP3 BDKRB1 623/4885AGTR1 190/4885AGTR2 210/4885
US-11718591-B2 Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2- methylpentanoic acid and uses thereof MME, CTSC, REN BDKRB1 1268/4885AGTR1 25/4885AGTR2 42/4885
US-20050288272-A1 Pharmaceutical compositions comprising NEP-inhibitors, inhibitors of the endogenous endothelin producing system and AT1 receptor antagonists ECE1, EDNRA, MME BDKRB1 132/4885AGTR1 6/4885AGTR2 7/4885
US-11851443-B2 Neprilysin inhibitors MME, REN, ACE BDKRB1 39/4885AGTR1 4/4885AGTR2 9/4885
US-12016835-B2 Neprilysin inhibitors MME, REN, ACE BDKRB1 41/4885AGTR1 5/4885AGTR2 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.