SCHEMBL16720656

SCHEMBL16720656

Fc1ccc(-n2ccc3cc[c]cc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.45
BIRC5 O15392 1/20 0.39
CYP19A1 P11511 2/20 0.36
ALDH1A1 P00352 5/20 0.33
KDM4E B2RXH2 4/20 0.33
MAPT P10636 4/20 0.33
HPGD P15428 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
RAB9A P51151 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP3A4 P08684 1/20 0.33
LMNA P02545 2/20 0.32
HTT P42858 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL148060 0.86 KCNH2 (0.49) KCNH2BIRC5CYP19A1ALDH1A1KDM4E
SCHEMBL16719505 0.83 BIRC5 (0.39) BIRC5CYP19A1ALDH1A1MAPTLMNA
SCHEMBL145426 0.82 BIRC5 (0.44) BIRC5CYP19A1SMN1; SMN2HTT
SCHEMBL16719992 0.81 HPGDS (0.36) KCNH2BIRC5MAPTCDC7CDK2
SCHEMBL16720593 0.79 CYP19A1 (0.45) BIRC5CYP19A1MAPTCDC7CDK2
SCHEMBL4273291 0.79 ALDH1A1 (0.39) BIRC5ALDH1A1KDM4EMAPTHPGD
SCHEMBL16719663 0.78 MAPT (0.34) KCNH2MAPTCDC7CDK2ROCK1
SCHEMBL16720871 0.78 POLB (0.39) BIRC5ALDH1A1KDM4EMAPTHPGD
SCHEMBL16720518 0.76 ROCK2 (0.43) BIRC5CYP19A1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL16720528 0.76 MAPT (0.42) BIRC5ALDH1A1KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed