SCHEMBL16748752

SCHEMBL16748752

CCCCOc1cn(OCCCC)c(CNO)cc1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.34
GAA P10253 3/20 0.34
TSHR P16473 3/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
CRHBP P24387 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
ATM Q13315 1/20 0.33
CRHR2 Q13324 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16748757 0.88 S1PR2 (0.33) TP53GAATSHRHTTTDP1
SCHEMBL9915355 0.85 COMT (0.38) TP53GAATDP1ALDH1A1L3MBTL1
SCHEMBL15279057 0.84 TP53 (0.33) TP53GAATSHRHTTTDP1
SCHEMBL9915322 0.82 CYP1A2 (0.34) TP53GAATSHRHTTTDP1
SCHEMBL9915436 0.80 FAAH (0.36) TSHRALDH1A1MAPK1
SCHEMBL9915493 0.80 SMN1; SMN2 (0.43) HPGDCASP1HSD17B10SMPD1KMT2A
SCHEMBL14136527 0.80 PPARD (0.43) TP53TSHRHPGDHSD17B10MAPT
SCHEMBL14136603 0.80 USP2 (0.45) MAPK1
SCHEMBL14136604 0.80 USP2 (0.45) GAAHPGDMAPK1SMPD1MAPT
SCHEMBL16748764 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646436-B1 MONOBACTAMS PFIZER (US) 2015-05-27 EP disclosed