SCHEMBL16795100

SCHEMBL16795100

CCOC(=O)n1cc(C(=O)c2ccccc2N)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
HSD17B10 Q99714 1/20 0.51
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.47
POLB P06746 1/20 0.47
CNR1 P21554 5/20 0.47
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
ESRRA P11474 1/20 0.44
CNR2 P34972 3/20 0.43
TSHR P16473 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.43
CREBBP Q92793 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16796720 0.86 MEN1 (0.43) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
SCHEMBL16796718 0.84 ALDH1A1 (0.46) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
SCHEMBL2117439 0.82 KMT2A (0.55) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2457012 0.81 KMT2A (0.64) ALDH1A1NPSR1MEN1KMT2AL3MBTL1
SCHEMBL2114760 0.76 L3MBTL1 (0.54) ALDH1A1MEN1KMT2AL3MBTL1POLB
SCHEMBL6283431 0.75 L3MBTL1 (0.53) ALDH1A1HSD17B10MEN1KMT2AL3MBTL1
SCHEMBL2544694 0.74 L3MBTL1 (0.52) ALDH1A1NPSR1MEN1KMT2AL3MBTL1
SCHEMBL15902156 0.72 ALDH1A1 (0.67) ALDH1A1MEN1KMT2AL3MBTL1POLB
SCHEMBL8560375 0.72 L3MBTL1 (0.67) ALDH1A1NPSR1MEN1KMT2AL3MBTL1
SCHEMBL9164757 0.71 L3MBTL1 (0.60) ALDH1A1HSD17B10MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088564-A1 P2X4 RECEPTOR MODULATING COMPOUNDS SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed