SCHEMBL16795366

SCHEMBL16795366

CC1(C)OB(c2ccc(CN3CCN(C(=O)O)CC3)c(O)c2)OC1(C)C

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.47
FAAH O00519 2/20 0.39
ALDH1A1 P00352 2/20 0.38
HIF1A Q16665 5/20 0.37
LIPG Q9Y5X9 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
MPO P05164 1/20 0.35
GRIN2B Q13224 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MGLL Q99685 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3416907 0.82 HRH3 (0.47) ALDH1A1LIPGMEN1KMT2A
SCHEMBL16795211 0.81 POLB (0.46) ROCK1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL3045151 0.80 LIPG (0.47) FAAHALDH1A1LIPGMEN1KMT2A
SCHEMBL17136271 0.77 DGAT1 (0.42) ROCK1FAAHALDH1A1KDM4E
SCHEMBL15094169 0.76 ROCK1 (0.51) ROCK1ALDH1A1KDM4EMGLL
SCHEMBL16795444 0.74 GRIN2B (0.38) GRIN2BKDM4E
SCHEMBL25207195 0.74 ROCK1 (0.54) ROCK1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL18579955 0.73 ROCK1 (0.53) ROCK1ALDH1A1LIPGMPOKDM4E
SCHEMBL16795231 0.73 ALDH1A1 (0.50) FAAHALDH1A1MEN1KMT2AMPO
SCHEMBL23111584 0.73 FAAH (0.55) FAAHALDH1A1MEN1KMT2AMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015086693-A1 PYRAZOLOPYRIMIDIN-2-YL DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2015-06-18 WO disclosed