SCHEMBL16796597

SCHEMBL16796597

O=C1CN=C(c2cccc(NS(=O)(=O)c3ccccc3)c2)c2[nH]c3ccccc3c2N1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.49
MMP9 P14780 1/20 0.49
MMP8 P22894 1/20 0.49
MMP13 P45452 1/20 0.49
BRD4 O60885 2/20 0.45
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
KDM1A O60341 2/20 0.41
POLB P06746 1/20 0.41
BRAF P15056 1/20 0.40
MAPT P10636 1/20 0.40
PDE4B Q07343 1/20 0.40
PFKFB3 Q16875 1/20 0.40
P2RX4 Q99571 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16796729 0.85 P2RX4 (0.43) ALDH1A1HPGDLMNAKMT2AMAPT
SCHEMBL16796607 0.82 P2RX4 (0.41) ALDH1A1KMT2AMAPTP2RX4
SCHEMBL16239013 0.82 P2RX4 (0.54) MMP2MMP9MMP8MMP13ALDH1A1
SCHEMBL16796643 0.81 METAP2 (0.44) ALDH1A1HPGDHTTMAPTP2RX4
SCHEMBL16812977 0.81 GABRA1 (0.51) ALDH1A1HPGDHTTLMNAMAPT
SCHEMBL16796629 0.80 KMT2A (0.50) MMP2MMP9MMP8MMP13BRD4
SCHEMBL16796688 0.79 P2RX4 (0.47) ALDH1A1HPGDHTTLMNAKMT2A
SCHEMBL16813006 0.78 P2RX4 (0.46) ALDH1A1HPGDLMNAKMT2AMEN1
SCHEMBL16796615 0.78 P2RX4 (0.46) ALDH1A1HPGDKMT2ATP53MAPT
SCHEMBL16796606 0.78 P2RX4 (0.46) ALDH1A1HPGDLMNAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed