SCHEMBL16796608

SCHEMBL16796608

COc1ccc(C2=NCC(=O)Nc3c2[nH]c2ccccc32)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
GSK3B P49841 5/20 0.43
CDK5 Q00535 5/20 0.43
CDK5R1 Q15078 5/20 0.43
CCNB2 O95067 4/20 0.43
CDK1 P06493 4/20 0.43
CCNB1 P14635 4/20 0.43
CCNB3 Q8WWL7 4/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16813010 0.92 ALDH1A1 (0.47) ALDH1A1CA1CA2CA4CA6
SCHEMBL16796630 0.86 CA1 (0.41) ALDH1A1CA1CA2CA4CA6
SCHEMBL16812997 0.83 GABRA1 (0.50) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL16812980 0.82 ALDH1A1 (0.52) ALDH1A1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL16812979 0.82 CHRM4 (0.59) ALDH1A1GSK3BCDK5CDK5R1CCNB2
SCHEMBL16796684 0.81 TLR8 (0.38) GSK3BCCNB2CDK1CCNB1CCNB3
SCHEMBL16796584 0.80 GABRA1 (0.38) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL16812999 0.80 GSK3B (0.44) ALDH1A1CA1CA2CA4CA6
SCHEMBL16813012 0.80 GSK3B (0.43) ALDH1A1CA1CA2CA4CA6
SCHEMBL16812971 0.80 ALDH1A1 (0.62) ALDH1A1GSK3BCDK5CDK5R1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed