SCHEMBL16812979

SCHEMBL16812979

COc1cccc(C2=NCC(=O)Nc3c2[nH]c2ccccc32)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.59
DRD2 P14416 2/20 0.59
HTR7 P34969 2/20 0.59
ALDH1A1 P00352 2/20 0.52
NR1I2 O75469 1/20 0.46
CYP1A2 P05177 1/20 0.46
VDR P11473 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2B6 P20813 1/20 0.46
AHR P35869 1/20 0.46
NR1I3 Q14994 1/20 0.46
SERPINE1 P05121 1/20 0.46
F2 P00734 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
P2RX4 Q99571 1/20 0.43
TUBB4A P04350 2/20 0.43
TUBB P07437 2/20 0.43
TUBA3C P0DPH7 2/20 0.43
TUBA1B P68363 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16796600 0.89 CHRM4 (0.46) CHRM4DRD2HTR7ALDH1A1CYP1A2
SCHEMBL16813014 0.89 CHRM4 (0.51) CHRM4DRD2HTR7ALDH1A1SERPINE1
SCHEMBL16813021 0.89 CHRM4 (0.51) CHRM4DRD2HTR7ALDH1A1NR1I2
SCHEMBL16812981 0.88 CHRM4 (0.46) CHRM4DRD2HTR7ALDH1A1NR1I2
SCHEMBL16812980 0.87 ALDH1A1 (0.52) CHRM4DRD2HTR7ALDH1A1HPGD
SCHEMBL16812971 0.87 ALDH1A1 (0.62) CHRM4DRD2HTR7ALDH1A1CYP1A2
SCHEMBL16813006 0.85 P2RX4 (0.46) CHRM4DRD2HTR7ALDH1A1CYP1A2
SCHEMBL16796604 0.84 P2RX4 (0.41) CHRM4DRD2HTR7ALDH1A1KMT2A
SCHEMBL16796688 0.84 P2RX4 (0.47) CHRM4DRD2HTR7ALDH1A1HPGD
SCHEMBL16812977 0.83 GABRA1 (0.51) ALDH1A1HPGDP2RX4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed