SCHEMBL1680715

SCHEMBL1680715

COc1ccc2cccccc1-2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 4/20 0.52
LMNA P02545 2/20 0.52
GAA P10253 1/20 0.52
PTPRC P08575 1/20 0.52
PTPN1 P18031 1/20 0.52
XDH P47989 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HSD17B10 Q99714 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
ACACA Q13085 1/20 0.49
NPC1 O15118 1/20 0.49
TP53 P04637 1/20 0.49
RAB9A P51151 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
APP P05067 1/20 0.48
USP2 O75604 1/20 0.48
MAPT P10636 1/20 0.48
DUSP3 P51452 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24106783 0.93 ALDH1A1 (0.55) ALDH1A1KDM4ELMNAGAAPTPRC
SCHEMBL294721 0.93 ALDH1A1 (0.58) ALDH1A1KDM4ELMNAGAAPTPRC
SCHEMBL30136447 0.93 ALDH1A1 (0.58) ALDH1A1KDM4ELMNAGAAPTPRC
Biphenyl SCHEMBL9989359 0.91 ALDH1A1 (0.56) ALDH1A1KDM4ELMNAGAAPTPRC
SCHEMBL30017788 0.91 ALDH1A1 (0.56) ALDH1A1KDM4ELMNAGAAPTPRC
Methyl Alcohol SCHEMBL28372647 0.88 ALDH1A1 (0.55) ALDH1A1KDM4ELMNAGAAPTPRC
Methylamine SCHEMBL28363123 0.88 ALDH1A1 (0.55) ALDH1A1KDM4ELMNAGAAPTPRC
SCHEMBL20550260 0.87 PTPRC (0.54) ALDH1A1KDM4ELMNAGAAPTPRC
SCHEMBL12326181 0.86 MAOA (0.53) ALDH1A1KDM4EPTPRCPTPN1MEN1
SCHEMBL27755757 0.86 SYK (0.56) ALDH1A1KDM4ELMNAGAAPTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837973-A Fragrance materials PROCTER & GAMBLE 2015-08-12 CN disclosed
US-20110195999-A1 NOVEL ANTIFUNGAL AGENT CONTAINING HETEROCYCLIC COMPOUND NAKAMOTO KAZUTAKA 2011-08-11 US disclosed
US-7932272-B2 Antifungal agent containing heterocyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-04-26 US disclosed
US-7829585-B2 Antifungal agent containing pyridine derivative EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-11-09 US disclosed
US-20090062348-A1 Antifungal Agent Containing Pyridine Derivative EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-03-05 US disclosed
EP-1864980-A1 ANTIFUNGAL AGENT CONTAINING PYRIDINE DERIVATIVE Eisai R&D Management Co., Ltd. (JP) 2007-12-12 EP disclosed
US-20070105943-A1 Novel antifungal agent containing heterocyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2007-05-10 US disclosed
US-7074798-B2 Xanthine derivative and DPPIV inhibitor EISAI CO., LTD (JP) 2006-07-11 US disclosed
EP-1669348-A1 NOVEL ANTIFUNGAL AGENT COMPRISING HETEROCYCLIC COMPOUND Eisai Co., Ltd. (JP) 2006-06-14 EP disclosed
EP-1338595-B1 Xanthine derivatives as DPP-IV inhibitors EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-20040082570-A1 Xanthine derivative and DPPIV inhibitor EISAI CO., LTD. (JP) 2004-04-29 US disclosed
EP-1338595-A2 Xanthine derivatives as DPP-IV inhibitors Eisai Co., Ltd. (JP) 2003-08-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082570-A1 Xanthine derivative and DPPIV inhibitor DPP4, DPP9, DPP7 ALDH1A1 112/4885KDM4E 1550/4885LMNA 4075/4885
US-20110195999-A1 NOVEL ANTIFUNGAL AGENT CONTAINING HETEROCYCLIC COMPOUND ERG28, CYP51A1, XPO1 ALDH1A1 1677/4885KDM4E 3112/4885LMNA 2372/4885
US-20070105943-A1 Novel antifungal agent containing heterocyclic compound ERG28, DPM1, CYP51A1 ALDH1A1 1459/4885KDM4E 3245/4885LMNA 2208/4885
US-20090062348-A1 Antifungal Agent Containing Pyridine Derivative ERG28, SQOR, CYP51A1 ALDH1A1 602/4885KDM4E 2090/4885LMNA 4768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.