SCHEMBL16813014

SCHEMBL16813014

COc1cccc(C2=NCC(=O)Nc3c2[nH]c2ccc(Cl)cc32)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.51
DRD2 P14416 2/20 0.51
HTR7 P34969 2/20 0.51
ALDH1A1 P00352 1/20 0.46
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
CNR1 P21554 1/20 0.41
NTSR1 P30989 1/20 0.41
OPRK1 P41145 1/20 0.41
PDE4D Q08499 1/20 0.41
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
GSK3B P49841 2/20 0.41
PRKCA P17252 1/20 0.41
STK10 O94804 1/20 0.40
SLK Q9H2G2 1/20 0.40
SERPINE1 P05121 1/20 0.39
TUBB4A P04350 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16812979 0.89 CHRM4 (0.59) CHRM4DRD2HTR7ALDH1A1GSK3B
SCHEMBL16813021 0.88 CHRM4 (0.51) CHRM4DRD2HTR7ALDH1A1LMNA
SCHEMBL16813036 0.85 CNR1 (0.56) ALDH1A1MAPTCNR1NTSR1OPRK1
SCHEMBL16796669 0.85 CNR1 (0.43) CNR1NTSR1OPRK1PDE4DGSK3B
SCHEMBL16812971 0.84 ALDH1A1 (0.62) CHRM4DRD2HTR7ALDH1A1MAPT
SCHEMBL16796592 0.83 PTGS2 (0.49) CNR1NTSR1OPRK1PDE4DGSK3B
SCHEMBL16812983 0.81 CNR1 (0.47) CHRM4DRD2HTR7MAPTLMNA
SCHEMBL16812975 0.81 GSK3B (0.45) CNR1NTSR1OPRK1PDE4DGSK3B
SCHEMBL16813009 0.80 GSK3B (0.43) LMNACNR1NTSR1OPRK1PDE4D
SCHEMBL16796600 0.78 CHRM4 (0.46) CHRM4DRD2HTR7ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed