SCHEMBL1684469

SCHEMBL1684469

Bc1cnc(N2CCC(C(N)=O)(c3ccccc3)CC2)nc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 3/20 0.52
OPRL1 P41146 2/20 0.47
OPRD1 P41143 5/20 0.44
HSD11B1 P28845 2/20 0.43
OPRM1 P35372 6/20 0.41
OPRK1 P41145 4/20 0.41
SLC22A1 O15245 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
KCNH2 Q12809 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
HDAC6 Q9UBN7 1/20 0.39
PTPN11 Q06124 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1282800 0.87 MLYCD (0.52) MLYCDOPRL1OPRD1HSD11B1OPRM1
SCHEMBL3422626 0.86 MLYCD (0.53) MLYCDOPRL1OPRD1HSD11B1OPRK1
SCHEMBL1684394 0.76 ALDH1A1 (0.38) OPRL1OPRD1OPRM1OPRK1HDAC6
SCHEMBL1282234 0.76 MLYCD (0.50) MLYCDOPRD1HSD11B1OPRM1OPRK1
SCHEMBL8366154 0.75 OPRL1 (0.56) MLYCDOPRL1OPRD1HSD11B1OPRM1
SCHEMBL2702494 0.73 OPRD1 (0.47) MLYCDOPRL1OPRD1KCNH2
SCHEMBL2702717 0.73 PKM (0.54) MLYCDOPRL1OPRD1
SCHEMBL1684410 0.73 MLYCD (0.49) MLYCDOPRL1OPRD1OPRM1
SCHEMBL2722547 0.73 AKR1C1 (0.57) MLYCDOPRL1OPRD1HSD11B1OPRM1
SCHEMBL501923 0.73 AKR1C1 (0.57) MLYCDOPRL1OPRD1HSD11B1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012045124-A1 BACTERIA TOPOISOMERASE II INHIBITING 2-ETHYLCARBAMOYLAMINO-1, 3-BENZOTHIAZOL-5-YLS BIOTA EUROPE LTD (GB) 2012-04-12 WO disclosed