SCHEMBL1685394

SCHEMBL1685394

CCNS(=O)(=O)c1cc(O)ccc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.51
BRD2 P25440 1/20 0.51
BRD3 Q15059 1/20 0.51
ALDH1A1 P00352 5/20 0.50
GAA P10253 3/20 0.50
TSHR P16473 2/20 0.50
LMNA P02545 2/20 0.49
HPGD P15428 1/20 0.49
HIF1A Q16665 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP3A4 P08684 1/20 0.47
RECQL P46063 1/20 0.47
MEP1B Q16820 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
GFER P55789 1/20 0.45
PKM P14618 1/20 0.44
HTT P42858 1/20 0.43
GLA P06280 1/20 0.42
HSD17B2 P37059 1/20 0.42
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834037 0.87 ALDH1A1 (0.48) BRD4BRD2BRD3ALDH1A1GAA
SCHEMBL8469458 0.84 CA12 (0.50) BRD4BRD2BRD3ALDH1A1GAA
SCHEMBL9005826 0.83 ALDH1A1 (0.54) BRD4BRD2BRD3ALDH1A1GAA
SCHEMBL17319218 0.82 SMN1; SMN2 (0.60) BRD4BRD2BRD3ALDH1A1GAA
SCHEMBL10913560 0.82 GAA (0.56) ALDH1A1GAATSHRLMNAHPGD
SCHEMBL9181456 0.82 RECQL (0.52) BRD4BRD2BRD3ALDH1A1GAA
SCHEMBL22409314 0.81 ALDH1A1 (0.48) ALDH1A1GAALMNAHPGDHIF1A
SCHEMBL758273 0.81 TSHR (0.48) BRD4BRD2BRD3ALDH1A1GAA
SCHEMBL743630 0.80 LMNA (0.65) BRD4ALDH1A1GAATSHRLMNA
SCHEMBL1032718 0.80 KDM4E (0.60) BRD4BRD2BRD3ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538070-B1 PHARMACEUTICAL COMPOSITION OF BENZENESULFONAMIDE DERIVATIVES FOR TREATMENT OF ADENOID CYSTIC CARCINOMA GONGWIN BIOPHARM CO LTD TAIWAN (TW) 2023-03-29 EP claimed
EP-3468547-B1 NOVEL BENZENESULFONAMIDE COMPOSITIONS FOR TREATMENT OF MALIGNANT PLEURAL EFFUSIONS GONGWIN BIOPHARM CO LTD TAIWAN (TW) 2021-10-06 EP claimed
EP-2606094-B1 SALT RESISTANT POLYAMIDE COMPOSITIONS DU PONT (US) 2017-02-01 EP claimed
EP-1943291-B1 HYDROLYSIS RESISTANT POLYAMIDE COMPOSITIONS, AND ARTICLES FORMED THEREFROM DU PONT (US) 2013-12-11 EP claimed
EP-1805442-B1 HYDROLYSIS RESISTANT POLYAMIDE COMPOSITIONS AND ARTICLES FORMED THEREFROM DU PONT (US) 2011-04-20 EP claimed
EP-1264212-B1 ELEMENTS FOR FORMING PRINT-OUT IMAGES DU PONT (US) 2009-02-18 EP claimed
EP-1389101-B1 TOLUENE SULFONAMIDE-CONTAINING ANTI-TUMOR COMPOSITION AND METHOD OF USE THEREOF PTS INTERNATIONAL INC (US) 2008-12-03 EP claimed
EP-1805264-B1 MARINE UMBILICAL COMPRISING HYDROLYSIS RESISTANT POLYAMIDES DU PONT (US) 2008-10-08 EP claimed
EP-0801663-B1 CURABLE SEALER AND/OR ADHESIVE COMPOSITION, METHOD FOR COATING SAME AND COATED SUBSTRATES MINNESOTA MINING & MFG (US) 1999-08-18 EP claimed
EP-0459304-B1 A one component sealant composition ADCO PRODUCTS INC (US) 1996-10-09 EP claimed
EP-0450105-B1 Room-temperature, moisture-curable, primerless, poluyrethane-based adhesive composition and method ADCO PRODUCTS INC (US) 1995-11-15 EP claimed
EP-0212135-B1 REMOISTENABLE HOT MELT ADHESIVES National Starch and Chemical Investment Holding Corporation (US) 1991-09-04 EP claimed
EP-0012521-B1 VESICULAR RECORDING MATERIALS AND PROCESS FOR THEIR PRODUCTION BEXFORD LIMITED (GB) 1983-03-23 EP claimed
US-8487016-B2 Dental impression material containing rheological modifiers and process of production 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-07-16 US disclosed
US-20110257290-A1 DENTAL IMPRESSION MATERIAL CONTAINING RHEOLOGICAL MODIFIERS AND PROCESS OF PRODUCTION 3M INNOVATIVE PROPERTIES COMPANY 2011-10-20 US disclosed
EP-2219585-A2 DENTAL IMPRESSION MATERIAL CONTAINING RHEOLOGICAL MODIFIERS AND PROCESS OF PRODUCTION 3M Innovative Properties Company (US) 2010-08-25 EP disclosed
EP-0553651-A1 Sulfonamides and their use DR. TH. BÖHME KG CHEM. FABRIK GMBH & CO. (DE) 1993-08-04 EP disclosed
EP-0006125-B1 PHOTOPOLYMERISABLE MIXTURE AND LIGHT-SENSITIVE COATING MATERIAL HOECHST AKTIENGESELLSCHAFT (DE) 1983-05-11 EP disclosed
EP-0035669-A2 Aqueous dispersions and process for making them BAYER AG (DE) 1981-09-16 EP disclosed
EP-0006125-A1 Photopolymerisable mixture and light-sensitive coating material HOECHST AKTIENGESELLSCHAFT (DE) 1980-01-09 EP disclosed