SCHEMBL1687290

SCHEMBL1687290

O=S(=O)(Nc1ccccc1B(O)O)c1cc(S(=O)(=O)c2ccccc2)cs1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GAB1 Q13480 1/20 0.45
MMP8 P22894 2/20 0.42
MMP3 P08254 1/20 0.42
CA2 P00918 5/20 0.40
ACLY P53396 2/20 0.40
HTR6 P50406 1/20 0.38
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21067285 0.80 ACLY (0.54) GAB1ACLY
SCHEMBL4316537 0.79 GAB1 (0.44) GAB1MMP8MMP3CA2HTR6
SCHEMBL14087505 0.78 GAB1 (0.51) GAB1MMP8MMP3CA2HTR6
SCHEMBL15880546 0.77 CA2 (0.52) GAB1MMP8MMP3CA2HTR6
SCHEMBL3556126 0.75 MEN1 (0.47) GAB1ACLYALDH1A1SMN1; SMN2
SCHEMBL13633850 0.74 SLC40A1 (0.65) ALDH1A1
SCHEMBL3552834 0.73 MEN1 (0.45) GAB1ACLYSMN1; SMN2
SCHEMBL7460372 0.73 HTR6 (0.56) GAB1MMP8MMP3CA2HTR6
SCHEMBL3557735 0.72 SLC16A3 (0.45) GAB1ACLYSMN1; SMN2
SCHEMBL3558197 0.72 SLC16A3 (0.60) GAB1ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2484680-A1 Useful Combinations of Monobactam Antibiotics with beta-Lac-tamase Inhibitors Basilea Pharmaceutica AG (CH) 2012-08-08 EP disclosed
EP-2308874-A1 Useful beta-lactamase inhibitors Basilea Pharmaceutica AG (CH) 2011-04-13 EP disclosed