SCHEMBL16888490

SCHEMBL16888490

Cc1c[n+]([O-])c(-c2cc(Cl)ccc2F)cc1Nc1cc[n+]([O-])cc1C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 7/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPK14 Q16539 1/20 0.38
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
BMPR1A P36894 1/20 0.33
ACVR1B P36896 1/20 0.33
ACVRL1 P37023 1/20 0.33
ACVR1 Q04771 1/20 0.33
MAPK1 P28482 1/20 0.33
CCR2 P41597 1/20 0.32
CCR9 P51686 1/20 0.32
MAP2K2 P36507 1/20 0.32
MAP2K1 Q02750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16888488 0.85 TGFBR1 (0.58) TGFBR1BMPR1AACVR1BACVRL1ACVR1
SCHEMBL16888489 0.83 TGFBR1 (0.55) TGFBR1CYP3A4BMPR1AACVR1BACVRL1
SCHEMBL18219788 0.79 MAPK14 (0.35) TGFBR1ALDH1A1MAPK14CYP3A4BMPR1A
SCHEMBL18219787 0.74 NUDT1 (0.47) TGFBR1BMPR1AACVR1BACVRL1ACVR1
SCHEMBL18221548 0.72 TGFBR1 (0.48) TGFBR1CYP3A4BMPR1AACVR1BACVRL1
SCHEMBL22270337 0.64 TGFBR1 (0.79) TGFBR1CYP3A4BMPR1AACVR1BACVRL1
SCHEMBL30294397 0.61 KDM4E (0.54) ALDH1A1KDM4EMAPK14
SCHEMBL22852993 0.61 KDM4E (0.54) ALDH1A1KDM4EMAPK14
SCHEMBL30564933 0.61 ALDH1A1 (0.56) ALDH1A1KDM4EGLAGAASMN1; SMN2
SCHEMBL910922 0.61 ALDH1A1 (0.56) ALDH1A1KDM4EGLAGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015103355-A1 COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-07-09 WO disclosed