SCHEMBL16892162

SCHEMBL16892162

NC(=O)CNCc1cccc(COc2ccc3c(c2)OCO3)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SPHK2 Q9NRA0 1/20 0.58
SPHK1 Q9NYA1 1/20 0.58
MAOB P27338 8/20 0.57
MAOA P21397 7/20 0.57
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
SCN3A Q9NY46 1/20 0.47
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16892218 0.90 SPHK2 (0.61) SPHK2SPHK1MAOBMAOANPC1
SCHEMBL16892157 0.82 SPHK2 (0.49) SPHK2SPHK1SCN3A
SCHEMBL16892177 0.82 MAOB (0.60) MAOBMAOANPC1RAB9A
SCHEMBL16892175 0.82 MAOB (0.60) MAOBMAOANPC1RAB9A
SCHEMBL8843511 0.80 DPP7 (0.59) NPC1RAB9AALDH1A1LMNATSHR
SCHEMBL16892226 0.80 ALDH1A1 (0.52) SPHK2SPHK1SCN3AALDH1A1MAPK1
SCHEMBL16892155 0.80 MAOB (0.52) MAOBMAOANPC1RAB9A
SCHEMBL16892201 0.80 MAOB (0.52) MAOBMAOANPC1RAB9A
Hydrochloric Acid SCHEMBL5009249 0.76 HEXA (0.52) MAOBMAOANPC1RAB9AALDH1A1
SCHEMBL964037 0.75 SPHK2 (0.67) SPHK2SPHK1MAOBMAOANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015101294-A1 COMPOUNDS WITH ANALGESIC ACTIVITY AND MEDICAL USE THEREOF 中国人民解放军军事医学科学院毒物药物研究所 2015-07-09 WO disclosed