SCHEMBL1697479

SCHEMBL1697479

O=CC(=O)c1ccccn1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.61
CES1 P23141 1/20 0.61
LMNA P02545 3/20 0.59
MAPT P10636 3/20 0.59
KDM4E B2RXH2 2/20 0.59
NPC1 O15118 2/20 0.59
PKM P14618 2/20 0.59
RAB9A P51151 2/20 0.59
L3MBTL1 Q9Y468 3/20 0.59
NAPRT Q6XQN6 1/20 0.59
P4HTM Q9NXG6 1/20 0.59
ALDH1A1 P00352 2/20 0.57
KMT2A Q03164 2/20 0.53
GSK3B P49841 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
GPR52 Q9Y2T5 1/20 0.51
MITF O75030 1/20 0.49
TP53 P04637 1/20 0.49
MEN1 O00255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6244793 0.81 ALDH1A1 (0.61) CES2CES1LMNAMAPTKDM4E
SCHEMBL13893380 0.81 CES2 (0.59) CES2CES1LMNAMAPTKDM4E
SCHEMBL585346 0.81 CES2 (0.59) CES2CES1LMNAMAPTKDM4E
SCHEMBL22462223 0.79 MAPT (0.66) CES2CES1LMNAMAPTKDM4E
SCHEMBL30668590 0.79 MAPT (0.66) CES2CES1LMNAMAPTKDM4E
SCHEMBL27621482 0.79 CES2 (0.69) CES2CES1LMNAMAPTKDM4E
SCHEMBL14305290 0.79 MAPT (0.61) CES2CES1LMNAMAPTKDM4E
SCHEMBL22478745 0.79 MAPT (0.61) CES2CES1LMNAMAPTKDM4E
SCHEMBL19787945 0.78 MAPT (0.64) CES2CES1LMNAMAPTKDM4E
SCHEMBL11334868 0.78 MAPT (0.69) CES2CES1LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 100 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108245518-A Utilize the method for two one for treating cancers of 3- (4- ((4- (morpholinomethyl) benzyl) oxygroup) -1- oxoisoindoline diindyl -2- bases) piperidines -2,6- 细胞基因公司 2018-07-06 CN claimed
CN-107935994-A The synthesis of 3 (5 amino, 2 methyl 4 oxoquinazolin 3 (4H) base) piperidines, 2,6 diketone 细胞基因公司 2018-04-20 CN claimed
CN-105377831-B Synthesis of 3- (5-amino-2-methyl-4-oxoquinazolin-3 (4H) -yl) piperidine-2, 6-dione 细胞基因公司 2018-02-02 CN claimed
CN-105209462-A Novel inhibitor compounds of phosphodiesterase type 10A ABBVIE DEUTSCHLAND 2015-12-30 CN claimed
WO-2003082824-A1 SYNTHESIS OF 2,6-DICARBONYLPYRIDINES BOULDER SCIENTIFIC COMPANY (US) 2003-10-09 WO claimed
WO-2026101698-A1 HEPCIDIN MIMETIC COMPOUNDS AND USES THEREOF PROTAGONIST THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
US-12522618-B2 Copper complexes for treatment of neurodegenerative disorders ALS THERAPY DEVELOPMENT INSTITUTE (US) 2026-01-13 US disclosed
CN-120005601-A Acidizing corrosion inhibitor for oil field and preparation method thereof 黑龙江克瑞休斯石油科技有限公司 2025-05-16 CN disclosed
US-20240368195-A1 COPPER COMPLEXES FOR TREATMENT OF NEURODEGENERATIVE DISORDERS ALS THERAPY DEVELOPMENT INST (US) 2024-11-07 US disclosed
US-12054472-B2 1,2,4-triazine-4-amine derivatives NXERA PHARMA UK LIMITED (GB) 2024-08-06 US disclosed
US-12012422-B2 Copper complexes for treatment of neurodegenerative disorders ALS THERAPY DEVELOPMENT INSTITUTE (US) 2024-06-18 US disclosed
EP-4204399-A1 COPPER COMPLEXES FOR TREATMENT OF NEURODEGENERATIVE DISORDERS ALS Therapy Development Institute (US) 2023-07-05 EP disclosed
US-5696240-A Macrocyclic complexes of yttrium, the lanthanides and the actinides having peripheral coupling functionalities VALLARINO LIDIA M (US) 1997-12-09 US disclosed
US-5480883-A Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-01-02 US disclosed
CN-1101038-A 4-substituted 6,9-bis(substituted-amino) benzo(g) isoquinoline-5, 10-Di-ones UNIV VERMONT (US) 1995-04-05 CN disclosed
US-5373093-A Macrocyclic complexes of yttrium, the lanthanides and the actinides having peripheral coupling functionalities NEWPORT INSTRUMENTS 1994-12-13 US disclosed
EP-0369000-A4 MACROCYCLIC COMPLEXES OF YTTRIUM, THE LANTHANIDES AND THE ACTINIDES HAVING PERIPHERAL COUPLING FUNCTIONALITIES 1993-06-02 EP disclosed
EP-0369000-A1 MACROCYCLIC COMPLEXES OF YTTRIUM, THE LANTHANIDES AND THE ACTINIDES HAVING PERIPHERAL COUPLING FUNCTIONALITIES Vallarino, Lidia M. (US) 1990-05-23 EP disclosed
WO-1989011868-A1 MACROCYCLIC COMPLEXES OF YTTRIUM, THE LANTHANIDES AND THE ACTINIDES HAVING PERIPHERAL COUPLING FUNCTIONALITIES COULTER ELECTRONICS, INC. (US) 1989-12-14 WO disclosed
EP-0225673-B1 PROCESS FOR THE PREPARATION OF ACYL UREAS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1989-10-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12012422-B2 Copper complexes for treatment of neurodegenerative disorders SOD1, SMN1; SMN2, CLN6 CES2 1672/4885CES1 4059/4885LMNA 1550/4885
US-12054472-B2 1,2,4-triazine-4-amine derivatives ADORA2A, ADORA2B, ADORA1 CES2 1506/4885CES1 1376/4885LMNA 1724/4885
US-20240368195-A1 COPPER COMPLEXES FOR TREATMENT OF NEURODEGENERATIVE DISORDERS SOD1, SMN1; SMN2, CLN6 CES2 1672/4885CES1 4059/4885LMNA 1550/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.