SCHEMBL17029337

SCHEMBL17029337

O=C(O)CN(CCO)Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
LMNA P02545 2/20 0.57
KCNH2 Q12809 1/20 0.55
TSHR P16473 1/20 0.50
POLB P06746 2/20 0.48
CRHBP P24387 2/20 0.48
CRHR2 Q13324 2/20 0.48
GAA P10253 2/20 0.45
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MMP1 P03956 2/20 0.44
MMP2 P08253 2/20 0.44
MMP9 P14780 2/20 0.44
MMP8 P22894 2/20 0.44
MMP13 P45452 2/20 0.44
CYP2C19 P33261 2/20 0.44
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
CYP1A2 P05177 1/20 0.42
NR1D1 P20393 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421520 0.91 KCNH2 (0.59) ALDH1A1LMNAKCNH2TSHRCRHBP
SCHEMBL8664094 0.90 KCNH2 (0.60) ALDH1A1LMNAKCNH2TSHRCRHBP
SCHEMBL4935242 0.88 ALDH1A1 (0.61) ALDH1A1LMNAKCNH2TSHRPOLB
SCHEMBL3148017 0.85 ALDH1A1 (0.76) ALDH1A1LMNATSHRPOLBCRHBP
SCHEMBL13014185 0.80 NR1D1 (0.66) ALDH1A1LMNAKCNH2TSHRPOLB
SCHEMBL15524258 0.80 CRHBP (0.59) ALDH1A1LMNATSHRPOLBCRHBP
SCHEMBL19491671 0.80 ALDH1A1 (0.65) ALDH1A1LMNAKCNH2TSHRPOLB
SCHEMBL3132717 0.79 HTT (0.53) ALDH1A1LMNATSHRGAAMAPT
SCHEMBL463691 0.79 KCNH2 (0.49) KCNH2POLBSMN1; SMN2SIGMAR1
SCHEMBL14129565 0.78 ALDH1A1 (0.52) ALDH1A1LMNAKCNH2TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9115094-B2 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using THE UNITED STATES OF AMERICA, NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS) (US) 2015-08-25 US disclosed