SCHEMBL13014185

SCHEMBL13014185

CC(C)(C)OC(=O)CN(CCO)Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 5/20 0.66
NR1H3 Q13133 1/20 0.53
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
MMP1 P03956 3/20 0.45
MMP2 P08253 3/20 0.45
MMP9 P14780 3/20 0.45
MMP8 P22894 3/20 0.45
MMP13 P45452 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
TSHR P16473 1/20 0.42
GAA P10253 1/20 0.42
POLB P06746 1/20 0.41
KCNH2 Q12809 2/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13014193 0.90 NR1D1 (0.66) NR1D1NR1H3ALDH1A1LMNAMMP1
SCHEMBL17029221 0.84 NR1D1 (0.65) NR1D1NR1H3ALDH1A1LMNAMMP1
SCHEMBL3844227 0.82 MEN1 (0.52) NR1D1NR1H3ALDH1A1LMNATSHR
SCHEMBL13014191 0.82 NR1D1 (0.56) NR1D1NR1H3ALDH1A1LMNAMMP1
SCHEMBL17029337 0.80 ALDH1A1 (0.57) NR1D1ALDH1A1LMNAMMP1MMP2
SCHEMBL3129212 0.80 NR1D1 (0.48) NR1D1ALDH1A1LMNAMMP1MMP2
SCHEMBL18633621 0.80 NR1D1 (0.62) NR1D1NR1H3ALDH1A1MMP1MMP2
SCHEMBL4935242 0.80 ALDH1A1 (0.61) ALDH1A1LMNASMN1; SMN2TSHRGAA
SCHEMBL25391995 0.79 NR1D1 (0.43) NR1D1NR1H3ALDH1A1LMNASMN1; SMN2
SCHEMBL17714014 0.78 ITGA4 (0.56) NR1D1NR1H3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9115094-B2 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using THE UNITED STATES OF AMERICA, NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS) (US) 2015-08-25 US disclosed
US-20100322855-A1 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2010-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100322855-A1 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using UACA, CLTC, PKD1 NR1D1 1424/4885NR1H3 2774/4885ALDH1A1 3456/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.