SCHEMBL1703357

SCHEMBL1703357

Nc1ccc(S(=O)(=O)c2ccc(N)cc2N)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.60
TSHR P16473 3/20 0.60
LMNA P02545 2/20 0.60
MPO P05164 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2C9 P11712 1/20 0.60
ALDH1A1 P00352 3/20 0.57
PKM P14618 2/20 0.57
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HKDC1 Q2TB90 1/20 0.47
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
USP2 O75604 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29480329 0.88 HTR6 (0.66) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL1162839 0.88 HTR6 (0.66) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL11021570 0.87 GAA (0.52) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL8143772 0.85 HTR6 (0.52) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL17774709 0.83 HTR6 (0.62) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL28506883 0.82 LMNA (0.68) HTR6TSHRLMNAALDH1A1PKM
SCHEMBL7189713 0.80 HSD11B1 (0.64) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL29388003 0.80 HTR6 (0.56) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL7190093 0.80 HTR6 (0.56) HTR6TSHRLMNAMPOCYP3A4
SCHEMBL7865326 0.80 HKDC1 (0.57) HTR6TSHRLMNAMPOCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4390596-A POLYAMINE, BIS-MALEIMIDE, FREE RADICAL CATALYST, FILLER RHONE-POULENC INDUSTRIES (FR) 1983-06-28 US claimed
US-4238591-A BIS-MALEIMIDE, SILANEDIOL OR SILOXANE RHONE-POULENC INDUSTRIES (FR) 1980-12-09 US claimed
US-4225498-A Preparation of N-substituted oligo-imides RHONE-POULENC INDUSTRIES (FR) 1980-09-30 US claimed
WO-2024043285-A1 RESIN COMPOSITION, COMPOSITE REINFORCING MATERIAL, MOLDED BODY, AND METHOD FOR RECOVERING REINFORCING FIBERS FROM COMPOSITE REINFORCING MATERIAL 旭化成株式会社 2024-02-29 WO disclosed
EP-2181211-B1 FIBERS COMPRISING COPOLYMERS CONTAINING STRUCTURES DERIVED FROM A PLURALITY OF AMINE MONOMERS INCLUDING 4,4' DIAMINO DIPHENYL SULFONE AND METHODS FOR MAKING SAME DU PONT (US) 2012-04-18 EP disclosed
EP-2181210-B1 FIBERS COMPRISING COPOLYMERS CONTAINING STRUCTURES DERIVED FROM 4.4' DIAMINO DIPHENYL SULFONE AND A PLURALITY OF ACID MONOMERS AND METHODS OF MAKING SAME DU PONT (US) 2010-12-01 EP disclosed
EP-2181211-A1 FIBERS COMPRISING COPOLYMERS CONTAINING STRUCTURES DERIVED FROM A PLURALITY OF AMINE MONOMERS INCLUDING 4,4' DIAMINO DIPHENYL SULFONE AND METHODS FOR MAKING SAME E. I. du Pont de Nemours and Company (US) 2010-05-05 EP disclosed
EP-2181210-A1 FIBERS COMPRISING COPOLYMERS CONTAINING STRUCTURES DERIVED FROM 4.4' DIAMINO DIPHENYL SULFONE AND A PLURALITY OF ACID MONOMERS AND METHODS OF MAKING SAME E. I. du Pont de Nemours and Company (US) 2010-05-05 EP disclosed
WO-2009026489-A1 FIBERS COMPRISING COPOLYMERS CONTAINING STRUCTURES DERIVED FROM 4.4' DIAMINO DIPHENYL SULFONE AND A PLURALITY OF ACID MONOMERS AND METHODS OF MAKING SAME E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-02-26 WO disclosed
WO-2009026490-A1 FIBERS COMPRISING COPOLYMERS CONTAINING STRUCTURES DERIVED FROM A PLURALITY OF AMINE MONOMERS INCLUDING 4,4' DIAMINO DIPHENYL SULFONE AND METHODS FOR MAKING SAME E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-02-26 WO disclosed
EP-0526490-B1 TEMPERATURE AND SOLVENT-RESISTANT INK FOR THE INK-JET PRINTING PROCESS BECK & CO AG DR (DE) 1994-07-20 EP disclosed
US-4012361-A Heat-stable polyimide resins from a bis-imide, a polyamine and an alazine RHONE-POULENC S.A. (FR) 1977-03-15 US disclosed
US-4010220-A AMINO COMPOUND, POLYURETHANE ELASTOMER RHONE-POULENC INDUSTRIES (FR) 1977-03-01 US disclosed
US-4005154-A Curing 1,2-epoxy with prepolymer based on polyamines and oligomers possessing imide groups RHONE-POULENC S.A. (FR) 1977-01-25 US disclosed
US-3998904-A POLYAMINES WITH IMIDE GROUPS RHONE-POULENC S.A. (FR) 1976-12-21 US disclosed
US-3978152-A HEAT-RESISTANT RESINS DERIVED FROM A BIS-IMIDE, AN EPOXY RESIN AND A POLYAMINE RHONE-POULENC INDUSTRIES (FR) 1976-08-31 US disclosed
US-3970714-A Heat-stable polyimide resin modified by unsaturated polyester RHONE-POULENC S.A. (FR) 1976-07-20 US disclosed
US-3966678-A Maleic anhydride-polyaldimine prepolymers RHONE-POULENC S.A. (FR) 1976-06-29 US disclosed
US-3950279-A DI- OR TRI-MALEIMIDE, AZOMETHINE, SOLID FOAMING AGENT CIBA-GEIGY CORPORATION (US) 1976-04-13 US disclosed
US-3947385-A Mixtures containing prepolymers, which can be converted to heat-resistant foamed plastics CIBA-GEIGY CORPORATION (US) 1976-03-30 US disclosed